Singlet oxygen in antimicrobial photodynamic therapy: photosensitizer-dependent production and decay in E. coli

Several families of photosensitizers are currently being scrutinized for antimicrobial photodynamic therapy applications. Differences in physical and photochemical properties can lead to different localization patterns as well as differences in singlet oxygen production and decay when the photosensi...

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Bibliographic Details
Authors: Nonell, Santi, Agut, Montserrat, Ragàs Amalrich, Xavier, He, Xin, Roxo-Rosa, Mónica, Rocha Gonsalves, António, Serra, Arménio C.
Format: article
Status:Published version
Publication Date:2013
Country:España
Institution:Varias* (Consorci de Biblioteques Universitáries de Catalunya, Centre de Serveis Científics i Acadèmics de Catalunya)
Repository:Recercat. Dipósit de la Recerca de Catalunya
OAI Identifier:oai:recercat.cat:20.500.14342/994
Online Access:http://hdl.handle.net/20.500.14342/994
https://doi.org/10.3390/molecules18032712
Access Level:Open access
Keyword:Fotoquimioteràpia
Anàlisi espectral
Escheríchia coli
Antimicrobial photodynamic therapy
Cationic photosensitizers
E. coli
Kinetics
Photodynamic inactivation
Singlet oxygen
Time-resolved near-IR spectroscopy
577
Description
Summary:Several families of photosensitizers are currently being scrutinized for antimicrobial photodynamic therapy applications. Differences in physical and photochemical properties can lead to different localization patterns as well as differences in singlet oxygen production and decay when the photosensitizers are taken up by bacterial cells. We have examined the production and fate of singlet oxygen in Escherichia coli upon photosensitization with three structurally-different cationic photosensitizers, namely New Methylene Blue N (NMB), a member of the phenothiazine family, ACS268, a hydrophobic porphyrin with a single cationic alkyl chain, and zinc(II)-tetramethyltetrapyridinoporphyrazinium salt, a phthalocyanine-like photosensitizer with four positive charges on the macrocycle core. The kinetics of singlet oxygen production and decay indicate different localization for the three photosensitizers, whereby NMB appears to localize in an aqueous-like microenvironment, whereas ACS268 localizes in an oxygen-shielded site, highly reactive towards singlet oxygen. The tetracationic zinc(II) tetrapyridinoporphyrazine is extensively aggregated in the bacteria and fails to produce any detectable singlet oxygen.