DETERMINATION OF THE CONFORMATIONSAND RELATIVE CONFIGURATIONS OF EXOCYCLIC AMINES

Knowledge of the absolute configuration and conformationof exocyclic amines is of great importance, particularly for compounds with biological activity. Also, determination ofthe stereoselectivity of a reaction is important for both the pharmaceutical and agricultural industries. The exocyclic amine...

Descripción completa

Detalles Bibliográficos
Autores: 173129, 173130, MONTALVO GONZALEZ, J. ASCENCION, INIESTRA GALINDO, MARIA GUADALUPE, ARIZA CASTOLO, ARMANDO
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2010
País:México
Institución:Universidad Autónoma de Nayarit
Repositorio:Repositorio Institucional Aramara de la UAN
Idioma:inglés
OAI Identifier:oai:dspace.uan.mx:123456789/1965
Acceso en línea:https://doi.org/10.1002/mrc.2693
http://dspace.uan.mx:8080/jspui/handle/123456789/1965
Access Level:acceso abierto
Palabra clave:1H
13C
15N RMN
conformación
configuración
amina exocíclica
conformation
configuration
exocyclic amine
MEDICINA Y CIENCIAS DE LA SALUD [3]
Descripción
Sumario:Knowledge of the absolute configuration and conformationof exocyclic amines is of great importance, particularly for compounds with biological activity. Also, determination ofthe stereoselectivity of a reaction is important for both the pharmaceutical and agricultural industries. The exocyclic amines are a key group of compounds because they are the source of many interesting substances in these industries. Some of the amines reported here have been used as chiral inductors, particularly the derivatives of 1-phenylethylamine and 1-(naphthalen-2-yl) ethylamine. The cyclohexanamines and their N-substituted derivatives form a group of secondary amines with a variety of basicities that can be used in the synthesis of complex molecules; currently, N-(propan-2-yl) cyclohexanamine is used as a base for the deprotonation of slightly acidic compounds through the preparation of a lithium amide.