Pan-BCL2 family inhibitor obatoclax as treatment for parental and cisplatin-resistant triple negative breast cancer

Triple negative breast cancer (TNBC) is an incurable disease where novel therapeutic strategies are needed. Nowadays, only chemotherapy and radi otherapy are standard treatments for TNBC. Cancer stem cells population (CSCs) are one of the most important mechanism to appear chemoresistance process. B...

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Detalles Bibliográficos
Autores: Noblejas López, María del Mar, Nuncia Cantarero, Miriam, Tebar García, D., López Rosa, Raquel, Nieto Jiménez, Cristina, Burgos, Miguel, Galán Moya, Eva María
Tipo de recurso: capítulo de libro
Fecha de publicación:2020
País:España
Institución:Universidad de Castilla-La Mancha
Repositorio:RUIdeRA. Repositorio Institucional de la UCLM
OAI Identifier:oai:ruidera.uclm.es:10578/30500
Acceso en línea:http://hdl.handle.net/10578/30500
Access Level:acceso abierto
Palabra clave:Triple negative breast cancer
Obatoclax
Cisplatin
Resistant
BCL2 family
Descripción
Sumario:Triple negative breast cancer (TNBC) is an incurable disease where novel therapeutic strategies are needed. Nowadays, only chemotherapy and radi otherapy are standard treatments for TNBC. Cancer stem cells population (CSCs) are one of the most important mechanism to appear chemoresistance process. BCL2 family proteins are involved in apoptosis. We hypothesized that they be engaged in acquisition of resistance mechanism to chemotherapy due to the alteration of this family in CSCs population. So, in this work, we explored the antitumoral activity of BCL2 family proteins inhibitors, specifi cally, obatoclax (a pan-BCL2 family proteins inhibitor) in TNBC cells and in a chemoresistant TNBC cell model.