Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity

The oxidation of aliphatic C-H bonds is a very powerful reaction because it allows the functionalization of inert C-H bonds, converting them into a suitable sites for further chemical elaboration. It also represents one of the most challenging reactions in modern synthetic organic chemistry because...

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Detalles Bibliográficos
Autor: Milan, Michela
Tipo de recurso: tesis doctoral
Estado:Versión publicada
Fecha de publicación:2018
País:España
Institución:CBUC, CESCA
Repositorio:TDR. Tesis Doctorales en Red
OAI Identifier:oai:www.tdx.cat:10803/664865
Acceso en línea:http://hdl.handle.net/10803/664865
Access Level:acceso abierto
Palabra clave:C-H oxidation
Oxidació de CH
Oxidación de CH
Manganeses complexes
Complexos de manganès
Complejos de manganeso
Bioinspired models
Models bioinspirats
Modelos bioinspirados
Metal catalysts
Catalitzadors de metalls
Catalizadores de metales
546
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spelling Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivityMilan, MichelaC-H oxidationOxidació de CHOxidación de CHManganeses complexesComplexos de manganèsComplejos de manganesoBioinspired modelsModels bioinspiratsModelos bioinspiradosMetal catalystsCatalitzadors de metallsCatalizadores de metales546The oxidation of aliphatic C-H bonds is a very powerful reaction because it allows the functionalization of inert C-H bonds, converting them into a suitable sites for further chemical elaboration. It also represents one of the most challenging reactions in modern synthetic organic chemistry because the multitude of aliphatic C-H bonds in a molecule makes site selective oxidation particularly difficult. Moreover, the introduction of chirality represents an unmet but very appealing challenge, because the asymmetric oxidation of hydrocarbons produces chiral compounds of high value in organic synthesis from readily available starting materials. Until now, examples of enantioselective oxidation of nonactivated aliphatic C-H bonds remain exclusive to enzymes. This thesis has been devoted to the development of new catalytic systems capable to oxidize nonactivated aliphatic C-H bonds in a site-selective and enantioselective manner. In particularly, chemo- and enantioselective aliphatic C-H oxidation reactions, especially focused in amide containing substrates have been developed.L'oxidació d’enllaços C-H alifàtics és una reacció altament interessant perquè permet funcionalitzar l'enllaç C-H inert, generant molècules d’alt interès sintètic. No obstant, també es tracta d'una de les reaccions que més atenció ha generat en en el camp de la química orgànica sintètica moderna perquè la multitud d'enllaços C-H alifàtics present en una mateixa molècula fa que l'oxidació selectiva d’un enllaç específic sigui particularment difícil. A més, la introducció de quiralitat en aquesta reacció representa, encara a dia d’avui, un repte molt atractiu, ja que l'oxidació asimètrica d'hidrocarburs, compostos altament abundants a la naturalesa, permet l'obtenció de compostos quirals d'alt valor en síntesi orgànica; i de moment, segueix sent una transformació exclusiva dels enzims. En particular, s'han desenvolupat reaccions d'oxidació de C-H alifàtiques quimio- i enantioselectives, enfocades en substrats que contenen un grup funcional amida.Universitat de GironaCostas Salgueiro, MiquelBietti, MassimoCostas Salgueiro, MiquelUniversitat de Girona. Departament de Química201920192018info:eu-repo/semantics/doctoralThesisinfo:eu-repo/semantics/publishedVersion340 p.application/pdfapplication/pdfapplication/pdfhttp://hdl.handle.net/10803/664865TDX (Tesis Doctorals en Xarxa)reponame:TDR. Tesis Doctorales en Redinstname:CBUC, CESCAInglésL'accés als continguts d'aquesta tesi queda condicionat a l'acceptació de les condicions d'ús establertes per la següent llicència Creative Commons: http://creativecommons.org/licenses/by/4.0/http://creativecommons.org/licenses/by/4.0/info:eu-repo/semantics/openAccessoai:www.tdx.cat:10803/6648652026-06-14T12:46:07Z
dc.title.none.fl_str_mv Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity
title Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity
spellingShingle Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity
Milan, Michela
C-H oxidation
Oxidació de CH
Oxidación de CH
Manganeses complexes
Complexos de manganès
Complejos de manganeso
Bioinspired models
Models bioinspirats
Modelos bioinspirados
Metal catalysts
Catalitzadors de metalls
Catalizadores de metales
546
title_short Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity
title_full Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity
title_fullStr Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity
title_full_unstemmed Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity
title_sort Oxidation of unactivated C-H bonds catalyzed by manganese complexes: control over site-selectivity and enantioselectivity
dc.creator.none.fl_str_mv Milan, Michela
author Milan, Michela
author_facet Milan, Michela
author_role author
dc.contributor.none.fl_str_mv Costas Salgueiro, Miquel
Bietti, Massimo
Costas Salgueiro, Miquel
Universitat de Girona. Departament de Química
dc.subject.none.fl_str_mv C-H oxidation
Oxidació de CH
Oxidación de CH
Manganeses complexes
Complexos de manganès
Complejos de manganeso
Bioinspired models
Models bioinspirats
Modelos bioinspirados
Metal catalysts
Catalitzadors de metalls
Catalizadores de metales
546
topic C-H oxidation
Oxidació de CH
Oxidación de CH
Manganeses complexes
Complexos de manganès
Complejos de manganeso
Bioinspired models
Models bioinspirats
Modelos bioinspirados
Metal catalysts
Catalitzadors de metalls
Catalizadores de metales
546
description The oxidation of aliphatic C-H bonds is a very powerful reaction because it allows the functionalization of inert C-H bonds, converting them into a suitable sites for further chemical elaboration. It also represents one of the most challenging reactions in modern synthetic organic chemistry because the multitude of aliphatic C-H bonds in a molecule makes site selective oxidation particularly difficult. Moreover, the introduction of chirality represents an unmet but very appealing challenge, because the asymmetric oxidation of hydrocarbons produces chiral compounds of high value in organic synthesis from readily available starting materials. Until now, examples of enantioselective oxidation of nonactivated aliphatic C-H bonds remain exclusive to enzymes. This thesis has been devoted to the development of new catalytic systems capable to oxidize nonactivated aliphatic C-H bonds in a site-selective and enantioselective manner. In particularly, chemo- and enantioselective aliphatic C-H oxidation reactions, especially focused in amide containing substrates have been developed.
publishDate 2018
dc.date.none.fl_str_mv 2018
2019
2019
dc.type.none.fl_str_mv info:eu-repo/semantics/doctoralThesis
info:eu-repo/semantics/publishedVersion
format doctoralThesis
status_str publishedVersion
dc.identifier.none.fl_str_mv http://hdl.handle.net/10803/664865
url http://hdl.handle.net/10803/664865
dc.language.none.fl_str_mv Inglés
language_invalid_str_mv Inglés
dc.rights.none.fl_str_mv http://creativecommons.org/licenses/by/4.0/
info:eu-repo/semantics/openAccess
rights_invalid_str_mv http://creativecommons.org/licenses/by/4.0/
eu_rights_str_mv openAccess
dc.format.none.fl_str_mv 340 p.
application/pdf
application/pdf
application/pdf
dc.publisher.none.fl_str_mv Universitat de Girona
publisher.none.fl_str_mv Universitat de Girona
dc.source.none.fl_str_mv TDX (Tesis Doctorals en Xarxa)
reponame:TDR. Tesis Doctorales en Red
instname:CBUC, CESCA
instname_str CBUC, CESCA
reponame_str TDR. Tesis Doctorales en Red
collection TDR. Tesis Doctorales en Red
repository.name.fl_str_mv
repository.mail.fl_str_mv
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score 15.300719