Synthesis of chiral carbosilane dendrimers with L-cysteine and N-acetyl-L-cysteine on their surface and their application as chiral selectors for enantiomer separation by capillary electrophoresis

The synthesis of chiral carbosilane dendrimers functionalized with cysteine and Nacetylcysteine groups is presented in this work. These dendrimers were obtained through thiol-ene addition reactions and their application as chiral selectors in Capillary Electrophoresis was investigated. Four drugs us...

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Detalles Bibliográficos
Autores: Quintana Sánchez, Sara|||0000-0003-3184-716X, Ortega Lopez, Paula|||0000-0003-0377-5429, Mata de la Mata, Francisco Javier de la|||0000-0003-0418-3935, Gómez Ramírez, Rafael|||0000-0001-6448-2414, Marina Alegre, María Luisa|||0000-0002-5583-1624, García González, María Ángeles|||0000-0001-6292-8232
Tipo de recurso: artículo
Fecha de publicación:2017
País:España
Institución:Universidad de Alcalá (UAH)
Repositorio:e_Buah Biblioteca Digital Universidad de Alcalá
Idioma:inglés
OAI Identifier:oai:ebuah.uah.es:10017/35870
Acceso en línea:http://hdl.handle.net/10017/35870
https://dx.doi.org/10.1016/j.tetasy.2017.10.028
Access Level:acceso abierto
Palabra clave:carbosilane
dendrimers
chiral
electrophoresis
Química
Chemistry
Descripción
Sumario:The synthesis of chiral carbosilane dendrimers functionalized with cysteine and Nacetylcysteine groups is presented in this work. These dendrimers were obtained through thiol-ene addition reactions and their application as chiral selectors in Capillary Electrophoresis was investigated. Four drugs used as model compounds were analyzed under different experimental conditions observing that the use of a first generation dendrimer containing 4 terminal N-Acetyl-L-cysteine groups enabled the enantiomeric discrimination of razoxane being this discrimination power similar to that obtained with other powerful chiral selectors such as cyclodextrins.