Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction

1,3,5-Trisubstituted tetramic acids and 2,3-disubstituted indole derivatives were prepared from β-keto esters derived from amino acids by their reaction with iodophenyl-2-trifluoroacetylamine under Cu-catalysis. Both heterocyclic systems were generated from the same starting materials by choice of t...

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Autores: García-Aranda, M. Isabel, García-López, M. Teresa, Pérez de Vega, M. Jesús, González-Muñiz, Rosario
Formato: artículo
Fecha de publicación:2014
País:España
Recursos:Consejo Superior de Investigaciones Científicas (CSIC)
Repositorio:DIGITAL.CSIC. Repositorio Institucional del CSIC
OAI Identifier:oai:digital.csic.es:10261/96241
Acesso em linha:http://hdl.handle.net/10261/96241
Access Level:acceso abierto
Palavra-chave:2,3-Disubstituted indoles
Tetramic acids
b-Keto esters
Amino acids
Diversity oriented synthesis
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spelling Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reactionGarcía-Aranda, M. IsabelGarcía-López, M. TeresaPérez de Vega, M. JesúsGonzález-Muñiz, Rosario2,3-Disubstituted indolesTetramic acidsb-Keto estersAmino acidsDiversity oriented synthesis1,3,5-Trisubstituted tetramic acids and 2,3-disubstituted indole derivatives were prepared from β-keto esters derived from amino acids by their reaction with iodophenyl-2-trifluoroacetylamine under Cu-catalysis. Both heterocyclic systems were generated from the same starting materials by choice of the appropriate reaction conditions. © 2013 Published by Elsevier Ltd.Peer Reviewed2014201420142014info:eu-repo/semantics/articlehttp://purl.org/coar/resource_type/c_6501http://hdl.handle.net/10261/96241reponame:DIGITAL.CSIC. Repositorio Institucional del CSICinstname:Consejo Superior de Investigaciones Científicas (CSIC)Inglésinfo:eu-repo/semantics/openAccessoai:digital.csic.es:10261/962412026-05-22T06:33:51Z
dc.title.none.fl_str_mv Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction
title Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction
spellingShingle Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction
García-Aranda, M. Isabel
2,3-Disubstituted indoles
Tetramic acids
b-Keto esters
Amino acids
Diversity oriented synthesis
title_short Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction
title_full Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction
title_fullStr Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction
title_full_unstemmed Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction
title_sort Tetramic acids and indole derivatives from amino acid β-keto esters. Fine-tuning the conditions of the key Cu-catalyzed reaction
dc.creator.none.fl_str_mv García-Aranda, M. Isabel
García-López, M. Teresa
Pérez de Vega, M. Jesús
González-Muñiz, Rosario
author García-Aranda, M. Isabel
author_facet García-Aranda, M. Isabel
García-López, M. Teresa
Pérez de Vega, M. Jesús
González-Muñiz, Rosario
author_role author
author2 García-López, M. Teresa
Pérez de Vega, M. Jesús
González-Muñiz, Rosario
author2_role author
author
author
dc.subject.none.fl_str_mv 2,3-Disubstituted indoles
Tetramic acids
b-Keto esters
Amino acids
Diversity oriented synthesis
topic 2,3-Disubstituted indoles
Tetramic acids
b-Keto esters
Amino acids
Diversity oriented synthesis
description 1,3,5-Trisubstituted tetramic acids and 2,3-disubstituted indole derivatives were prepared from β-keto esters derived from amino acids by their reaction with iodophenyl-2-trifluoroacetylamine under Cu-catalysis. Both heterocyclic systems were generated from the same starting materials by choice of the appropriate reaction conditions. © 2013 Published by Elsevier Ltd.
publishDate 2014
dc.date.none.fl_str_mv 2014
2014
2014
2014
dc.type.none.fl_str_mv info:eu-repo/semantics/article
http://purl.org/coar/resource_type/c_6501
format article
dc.identifier.none.fl_str_mv http://hdl.handle.net/10261/96241
url http://hdl.handle.net/10261/96241
dc.language.none.fl_str_mv Inglés
language_invalid_str_mv Inglés
dc.rights.none.fl_str_mv info:eu-repo/semantics/openAccess
eu_rights_str_mv openAccess
dc.source.none.fl_str_mv reponame:DIGITAL.CSIC. Repositorio Institucional del CSIC
instname:Consejo Superior de Investigaciones Científicas (CSIC)
instname_str Consejo Superior de Investigaciones Científicas (CSIC)
reponame_str DIGITAL.CSIC. Repositorio Institucional del CSIC
collection DIGITAL.CSIC. Repositorio Institucional del CSIC
repository.name.fl_str_mv
repository.mail.fl_str_mv
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