Dopamine induces intracellular Ca2+ signals mediated by alpha(1B)-adrenoceptors in rat pineal cells

We have studied the functional interaction of dopamine with a -adrenoceptor subtypes by measuring intracellular Ca2q 1 levels in pineal cells, a cell type where adrenoceptors are well characterized. We show that dopamine induces transient intracellular Ca2q signals in only 70% of cells responding to...

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Detalhes bibliográficos
Autores: Rey, Elkin, Hernández-Díaz, Francisco J., Abreu, Pedro, Alonso, Rafael, Tabares, Lucía
Formato: artículo
Estado:Versión publicada
Fecha de publicación:2001
País:España
Recursos:Universidad de Sevilla (US)
Repositorio:idUS. Depósito de Investigación de la Universidad de Sevilla
OAI Identifier:oai:idus.us.es:11441/146635
Acesso em linha:https://hdl.handle.net/11441/146635
https://doi.org/10.1016/S0014-2999(01)01250-X
Access Level:acceso abierto
Palavra-chave:Dopamine
α-Adrenoceptor
Pineal cell
Catecholamine
Descrição
Resumo:We have studied the functional interaction of dopamine with a -adrenoceptor subtypes by measuring intracellular Ca2q 1 levels in pineal cells, a cell type where adrenoceptors are well characterized. We show that dopamine induces transient intracellular Ca2q signals in only 70% of cells responding to phenylephrine. Dopamine-induced Ca2q signals desensitise faster than Ca2q transients elicited with phenylephrine and are selectively blocked by desipramine, imipramine, and a -adrenoceptor antagonists. These results suggest that 1B dopamine induced Ca2q signals are mainly due to the activation of one subtype of a-adrenoceptor, the a .