Synthesis of Analogues of Thyroid Hormones: Nuclear Receptor Modulators

Thyroid hormones are essential for the development and differentiation of all cells of the human body. This work reports the synthesis of some synthetic structural analogues of thyroid hormones, which may be modulators of the thyroid hormone receptor. The known compounds GC-1 (Sobe...

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Detalles Bibliográficos
Autores: de Castro, Guilherme Vieira, Rocha, Carlos Murilo Romero, Sanches, Vitor Lacerda, Ribeiro, Pedro H. Zana, Donate, Paulo Marcos, de Laurentiz, Rosangela da Silva, Polikarpov, Igor, Sairre, Mirela Ines
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2015
País:Brasil
Institución:Universidade Federal de Mato Grosso do Sul (UFMS)
Repositorio:Orbital - The Electronic Journal of Chemistry (Campo Grande)
Idioma:inglés
OAI Identifier:oai:periodicos.ufms.br:article/17872
Acceso en línea:https://periodicos.ufms.br/index.php/orbital/article/view/17872
Access Level:acceso abierto
Palabra clave:thyroid hormones
nuclear receptor
ligands
synthesis
Descripción
Sumario:Thyroid hormones are essential for the development and differentiation of all cells of the human body. This work reports the synthesis of some synthetic structural analogues of thyroid hormones, which may be modulators of the thyroid hormone receptor. The known compounds GC-1 (Sobetirome) and CG-24 were successfully prepared and two novel analogous molecules were also synthesized by a new and efficient synthetic methodology. DOI: http://dx.doi.org/10.17807/orbital.v7i3.739