Drug-conjugated monoclonal antibodies in advanced/metastatic breast cancer

The goal of this report is to analyze, in a general way, the structure and mechanism of action of drug-conjugated monoclonal (ADC) and examine the studies that led their approval in advanced/metastatic breast cancer (ABC). PubMed, Scopus and SciELO databases were used between 2000 and 2022; Bibliogr...

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Detalhes bibliográficos
Autores: Aldecoa-Bedoya, Franklin, Falcón, Silvia
Tipo de documento: artigo
Estado:Versão publicada
Data de publicação:2023
País:Perú
Recursos:Fundación Instituto Hipólito Unanue
Repositório:Diagnóstico
Idioma:espanhol
OAI Identifier:oai:revistadiagnostico.fihu.org.pe:article/427
Acesso em linha:https://revistadiagnostico.fihu.org.pe/index.php/diagnostico/article/view/427
Access Level:Acceso aberto
Palavra-chave:Anticuerpos monoclonales
inmunoconjugados
cáncer de mama
citostáticos
Antibody drug conjugates
antibodies
monoclonal
breast cancer
cytostatic agents
Descrição
Resumo:The goal of this report is to analyze, in a general way, the structure and mechanism of action of drug-conjugated monoclonal (ADC) and examine the studies that led their approval in advanced/metastatic breast cancer (ABC). PubMed, Scopus and SciELO databases were used between 2000 and 2022; Bibliographic references were searched for the keywords associated with ADC and ABC. ADCs combine classical monoclonal assays with a linker and a cytotoxic payload to destroy cancer cells in a targeted manner, when there is internalization of the corresponding receptor. There are currently three ACDs that have been approved for the treatment of CMAM; studies that have demonstrated significant advantages in progression-free survival when compared to standard treatment; evaluation of its main adverse events; implications for its management in our everyday lives; and potential inclusion in the current treatment of CMAM.