Role and New Insights of Pirfenidone in Fibrotic Diseases

Pirfenidone (PFD) is a non-peptide synthetic molecule issued as a broad-spectrum anti-fibrotic drug with the ability to decrease TGF-β1, TNF-α, PDGF and COL1A1 expression, which is highly related to prevent or remove excessive deposition of scar tissue in several organs. Basic and clinical evidence...

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Detalles Bibliográficos
Autores: Lopez de la Mora, David Alejandro, Sánchez Roque, Cibeles, Montoya Buelna, Margarita, Sánchez Enríquez, Sergio, Lucano Landeros, Silvia, Macias Barragan, José, Armendáriz Borunda, Juan Socorro
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2015
País:México
Institución:Universidad de Guadalajara
Repositorio:Repositorio UDG CUALTOS
OAI Identifier:oai:repositorio.cualtos.udg.mx:123456789/939
Acceso en línea:http://repositorio.cualtos.udg.mx:8080/jspui/handle/123456789/939
Access Level:acceso abierto
Palabra clave:pirfenidone
fibrosis
inflammation
idiopathic pulmonary fibrosis
Descripción
Sumario:Pirfenidone (PFD) is a non-peptide synthetic molecule issued as a broad-spectrum anti-fibrotic drug with the ability to decrease TGF-β1, TNF-α, PDGF and COL1A1 expression, which is highly related to prevent or remove excessive deposition of scar tissue in several organs. Basic and clinical evidence suggests that PFD may safely slow or inhibit the progressive fibrosis swelling after tissue injuries. Furthermore, a number of evidence suggests that this molecule will have positive effects in the treatment of other inflammatory diseases. This review contains current research in which PFD has been used as the treatment of several diseases, and focus mainly in the outcomes related to improve inflammation and fibrogenesis. Therefore, the main goal of this review is to focus on the novel findings of PFD efficacy rather than deepen in the chemical aspects of the molecule.