Constituents from Tithonia diversifolia. Stereochemical Revision of 2&-Hydroxytirotundin

A chemical study of the aerial parts of Tithonia diversifolialed to the isolation and stereostructural characterization of tagitininsA (1), C (2) and F (3), and a mixture of sterols. Tagitinin A (1) underwentspontaneous dehydration to 4 during the course of its 1H NMRmeasurement in CDCl3. The stereo...

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Detalles Bibliográficos
Autores: Abraham García, Guillermo Delgado
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2006
País:México
Institución:Universidad Nacional Autónoma de México
Repositorio:Redalyc-UNAM
OAI Identifier:oai:redalyc.org:47550407
Acceso en línea:https://www.redalyc.org/articulo.oa?id=47550407
Access Level:acceso abierto
Palabra clave:Química
2&#945
Tagitinins
furanheliangolides
Tithonia diversifolia
sesquiterpene lactones
Descripción
Sumario:A chemical study of the aerial parts of Tithonia diversifolialed to the isolation and stereostructural characterization of tagitininsA (1), C (2) and F (3), and a mixture of sterols. Tagitinin A (1) underwentspontaneous dehydration to 4 during the course of its 1H NMRmeasurement in CDCl3. The stereochemical analysis of 2α-hydroxytirotundin(5), an isomer of 1 previously reported by Kinghorn et al,led to the correction of its 3S,10S configuration to the 3S,10R stereochemistry.In addition, bioactivity evaluation of isolates showed themto exhibit moderate anti-inflammatory and cytotoxic activity