4-Amino-1,2,4-triazole-3-thione as a Promising Scaffold for the Inhibition of Serine and Metallo-β-Lactamases

© 2020 by the authors.

Bibliographic Details
Authors: Linciano, Pasquale, Gianquinto, Eleonora, Montanari, Martina, Maso, Lorenzo, Bellio, Pierangelo, Cebrián-Sastre, E., Celenza, Giuseppe, Blázquez, Jesús, Cendron, Laura, Spyrakis, Francesca, Tondi, Donatella
Format: article
Status:Published version
Publication Date:2020
Country:España
Institution:Consejo Superior de Investigaciones Científicas (CSIC)
Repository:DIGITAL.CSIC. Repositorio Institucional del CSIC
OAI Identifier:oai:digital.csic.es:10261/205617
Online Access:http://hdl.handle.net/10261/205617
Access Level:Open access
Keyword:4-amino-1,2,4-triazole-3-thione
Bacterial resistance
Structure-based drug design
Non-covalent inhibition
Thione/thiol tautomerism
Broad-spectrum activity
Description
Summary:© 2020 by the authors.