Advances toward a norovirus antiviral: from classical inhibitors to lethal mutagenesis

Human noroviruses are a leading cause of gastroenteritis worldwide, yet there are no licensed antivirals. There is an urgent need for norovirus therapeutics, particularly for chronic infections in immunocompromised individuals, but also a potential need for prophylactic use in epidemics. Continued r...

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Detalles Bibliográficos
Autores: Thorne , Lucy, Arias Esteban, Armando, Goodfellow , Ian
Tipo de recurso: artículo
Fecha de publicación:2016
País:España
Institución:Universidad de Castilla-La Mancha
Repositorio:RUIdeRA. Repositorio Institucional de la UCLM
OAI Identifier:oai:ruidera.uclm.es:10578/46895
Acceso en línea:https://hdl.handle.net/10578/46895
Access Level:acceso abierto
Palabra clave:Antivirals
Favipiravir
Human norovirus
Interferon
Lethal mutagenesis
Polymerase
Protease
Descripción
Sumario:Human noroviruses are a leading cause of gastroenteritis worldwide, yet there are no licensed antivirals. There is an urgent need for norovirus therapeutics, particularly for chronic infections in immunocompromised individuals, but also a potential need for prophylactic use in epidemics. Continued research has led to the identification of compounds that inhibit norovirus replication in vitro and, at least in some cases, are also effective in vivo against murine norovirus. Progress has included classical approaches targeting viral proteins and harnessing the antiviral action of interferon, strategies targeting essential host cell factors, and novel strategies exploiting the high mutation rate of noroviruses.