Mg/Fe-LDH: An efficient promoter for the synthesis of tetrahydrospiro[pyrazole-4,5′-pyrazolo[3,4-b]pyridine] derivatives

The synthesis of tetrahydrospiro[pyrazole-4,5'-pyrazolo[3,4-b]pyridine] derivativesusing Mg/Fe-LDH as a heterogeneous catalyst was reported. This methodology usedfor the condensation of pyrazolones with aldehydes in a basic medium and with thepresence of the Mg/Al-LDH catalyst presents many ben...

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Detalles Bibliográficos
Autores: Hibot, Achraf, Fadili, Hicham, Hafid, Abderrafia, Lebreton, Jacques, Pujol, Maria Dolors, Khouili, Mostafa
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2024
País:España
Institución:Universidad de Barcelona
Repositorio:Dipòsit Digital de la UB
OAI Identifier:oai:diposit.ub.edu:2445/224935
Acceso en línea:https://hdl.handle.net/2445/224935
Access Level:acceso abierto
Palabra clave:Metal·loporfirines
Química heterocíclica
Metalloporphyrines
Heterocyclic chemistry
Descripción
Sumario:The synthesis of tetrahydrospiro[pyrazole-4,5'-pyrazolo[3,4-b]pyridine] derivativesusing Mg/Fe-LDH as a heterogeneous catalyst was reported. This methodology usedfor the condensation of pyrazolones with aldehydes in a basic medium and with thepresence of the Mg/Al-LDH catalyst presents many benefits, such as the fact of using areusable and low-cost catalyst, environmentally friendly conditions, time short reactiontimes and excellent yields. It has been verified and confirmed that the catalyst isrelatively stable and allows its reuse without additional treatment. Condensation hasbeen carried out with different aldehydes and bis-pyrazolone derivatives have beenobtained with yields ranging from 71 to 91% of purified product. The stereo impedanceof the adduct formed prevents subsequent condensation.