Pharmacogenetics of ugt genes in North African populations

Cytochrome P450 (CYP450), sulfotransferase (SULT), and glucuronidase (UGT) enzymes play roles in the phase I and phase II metabolism of most clinically prescribed drugs. As polymorphisms in these genes may alter enzyme activities, most prescribed drugs will differ in their efficacy and side effects....

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Detalhes bibliográficos
Autores: Gaibar, M., Novillo, A., Romero-Lorca, A., Esteban i Torné, Maria Esther, Fernández-Santander, A.
Formato: artículo
Estado:Versión publicada
Fecha de publicación:2018
País:España
Recursos:Universidad de Barcelona
Repositorio:Dipòsit Digital de la UB
OAI Identifier:oai:diposit.ub.edu:2445/133582
Acesso em linha:https://hdl.handle.net/2445/133582
Access Level:acceso abierto
Palavra-chave:Enzims
Àfrica del Nord
Farmacogenètica
Enzymes
North Africa
Pharmacogenetics
Descrição
Resumo:Cytochrome P450 (CYP450), sulfotransferase (SULT), and glucuronidase (UGT) enzymes play roles in the phase I and phase II metabolism of most clinically prescribed drugs. As polymorphisms in these genes may alter enzyme activities, most prescribed drugs will differ in their efficacy and side effects. In prior work, we showed that besides polymorphisms in CYP450, those in SULT and UGT also give rise to different serum levels of some drug metabolites than detected in wild-type carriers of the genes [1]. [...]