Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy

[EN] Simple Summary Cancer is still the leading cause of disease-related death in pediatric populations and an important source of morbidity. These can be due to the neoplasm itself but also to the treatment administered; infants are patients of special vulnerability. The aim of this work was to ide...

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Autores: Urtasun, Andrea, Olivera, Gladys G., Sendra, Luis, Aliño, Salvador F., Berlanga, Pablo, Gargallo, Pablo, Balaguer, Julia, Juan-Ribelles, Antonio, Andrés, María del Mar, Cañete, Adela, Herrero, María José, Hervás-Marín, David|||0000-0003-0635-4961
Formato: artículo
Fecha de publicación:2023
País:España
Recursos:Universitat Politècnica de València (UPV)
Repositorio:RiuNet. Repositorio Institucional de la Universitat Politécnica de Valéncia
Idioma:inglés
OAI Identifier:oai:riunet.upv.es:10251/203844
Acesso em linha:https://riunet.upv.es/handle/10251/203844
Access Level:acceso abierto
Palavra-chave:Pharmacogenetics
SNP (single nucleotide polymorphism)
Chemotherapy
Infant
Toxicity
Therapeutic efficacy
Overall survival
Event-free survival
Anemia
Neutropenia
Thrombocytopenia
ESTADISTICA E INVESTIGACION OPERATIVA
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oai_identifier_str oai:riunet.upv.es:10251/203844
network_acronym_str ES
network_name_str España
repository_id_str
dc.title.none.fl_str_mv Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy
title Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy
spellingShingle Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy
Urtasun, Andrea
Pharmacogenetics
SNP (single nucleotide polymorphism)
Chemotherapy
Infant
Toxicity
Therapeutic efficacy
Overall survival
Event-free survival
Anemia
Neutropenia
Thrombocytopenia
ESTADISTICA E INVESTIGACION OPERATIVA
title_short Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy
title_full Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy
title_fullStr Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy
title_full_unstemmed Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy
title_sort Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to Chemotherapy
dc.creator.none.fl_str_mv Urtasun, Andrea
Olivera, Gladys G.
Sendra, Luis
Aliño, Salvador F.
Berlanga, Pablo
Gargallo, Pablo
Balaguer, Julia
Juan-Ribelles, Antonio
Andrés, María del Mar
Cañete, Adela
Herrero, María José
Hervás-Marín, David|||0000-0003-0635-4961
author Urtasun, Andrea
author_facet Urtasun, Andrea
Olivera, Gladys G.
Sendra, Luis
Aliño, Salvador F.
Berlanga, Pablo
Gargallo, Pablo
Balaguer, Julia
Juan-Ribelles, Antonio
Andrés, María del Mar
Cañete, Adela
Herrero, María José
Hervás-Marín, David|||0000-0003-0635-4961
author_role author
author2 Olivera, Gladys G.
Sendra, Luis
Aliño, Salvador F.
Berlanga, Pablo
Gargallo, Pablo
Balaguer, Julia
Juan-Ribelles, Antonio
Andrés, María del Mar
Cañete, Adela
Herrero, María José
Hervás-Marín, David|||0000-0003-0635-4961
author2_role author
author
author
author
author
author
author
author
author
author
author
dc.contributor.none.fl_str_mv Departamento de Estadística e Investigación Operativa Aplicadas y Calidad
Escuela Politécnica Superior de Alcoy
Escuela Técnica Superior de Ingeniería Agronómica y del Medio Natural
Asociación Pablo Ugarte
Instituto de Salud Carlos III
Repositorio Institucional de la Universitat Politècnica de València Riunet
dc.subject.none.fl_str_mv Pharmacogenetics
SNP (single nucleotide polymorphism)
Chemotherapy
Infant
Toxicity
Therapeutic efficacy
Overall survival
Event-free survival
Anemia
Neutropenia
Thrombocytopenia
ESTADISTICA E INVESTIGACION OPERATIVA
topic Pharmacogenetics
SNP (single nucleotide polymorphism)
Chemotherapy
Infant
Toxicity
Therapeutic efficacy
Overall survival
Event-free survival
Anemia
Neutropenia
Thrombocytopenia
ESTADISTICA E INVESTIGACION OPERATIVA
description [EN] Simple Summary Cancer is still the leading cause of disease-related death in pediatric populations and an important source of morbidity. These can be due to the neoplasm itself but also to the treatment administered; infants are patients of special vulnerability. The aim of this work was to identify genetic variants that correlate with significant impacts on treatments' safety and efficacy. 64 oncologic infant patients (under 18 months of age) were genotyped, calling for SNPs (single nucleotide polymorphisms) in genes related to the efficacy and/or toxicity of the chemotherapeutic drugs employed. The relationship of these genetic variants with 37 clinical parameters during 578 chemotherapy cycles was analyzed. Associations were found between 46 SNPs (in genes involved in drug transport and metabolism, gene repair, tumor suppression, and other biological functions) and survival and hematological toxicity. Following studies that confirm these findings, personalized medicine could be offered to improve response and tolerance to chemotherapeutic schemes. Background: Pharmacogenetics is a personalized medicine tool that aims to optimize treatments by adapting them to each individual's genetics, maximizing their efficacy while minimizing their toxicity. Infants with cancer are especially vulnerable, and their co-morbidities have vital repercussions. The study of their pharmacogenetics is new in this clinical field. Methods: A unicentric, ambispective study of a cohort of infants receiving chemotherapy (from January 2007 to August 2019). The genotypes of 64 patients under 18 months of age were correlated with severe drug toxicities and survival. A pharmacogenetics panel was configured based on PharmGKB, drug labels, and international experts' consortiums. Results: Associations between SNPs and hematological toxicity were found. Most meaningful were: MTHFR rs1801131 GT increasing the anemia risk (OR 1.73); rs1517114 GC, XPC rs2228001 GT, increasing neutropenia risk (OR 1.50 and 4.63); ABCB1 rs1045642 AG, TNFRSF11B rs2073618 GG, CYP2B6 rs4802101 TC and SOD2 rs4880 GG increasing thrombocytopenia risk (OR 1.70, 1.77, 1.70, 1.73, respectively). Regarding survival, MTHFR rs1801133 GG, TNFRSF11B rs2073618 GG, XPC rs2228001 GT, CYP3A4 rs2740574 CT, CDA rs3215400 del.del, and SLC01B1 rs4149015 GA were associated with lower overall survival probabilities (HR 3.12, 1.84, 1.68, 2.92, 1.90, and 3.96, respectively). Lastly, for event-free survival, SLC19A1 rs1051266 TT and CDA rs3215400 del.del increased the relapse probability (HR 1.61 and 2.19, respectively). Conclusions: This pharmacogenetic study is a pioneer in dealing with infants under 18 months of age. Further studies are needed to confirm the utility of the findings in this work to be used as predictive genetic biomarkers of toxicity and therapeutic efficacy in the infant population. If confirmed, their use in therapeutic decisions could improve the quality of life and prognosis of these patients.
publishDate 2023
dc.date.none.fl_str_mv 2023
2023-03-01
dc.type.none.fl_str_mv journal article
http://purl.org/coar/resource_type/c_6501
VoR
http://purl.org/coar/version/c_970fb48d4fbd8a85
dc.type.openaire.fl_str_mv info:eu-repo/semantics/article
format article
dc.identifier.none.fl_str_mv https://riunet.upv.es/handle/10251/203844
url https://riunet.upv.es/handle/10251/203844
dc.language.none.fl_str_mv Inglés
eng
language_invalid_str_mv Inglés
language eng
dc.relation.none.fl_str_mv Instituto de Salud Carlos III https://doi.org/10.13039/501100004587 IMP%2F00009
dc.rights.none.fl_str_mv open access
http://purl.org/coar/access_right/c_abf2
Reconocimiento (by)
http://creativecommons.org/licenses/by/4.0/
dc.rights.openaire.fl_str_mv info:eu-repo/semantics/openAccess
rights_invalid_str_mv open access
http://purl.org/coar/access_right/c_abf2
Reconocimiento (by)
http://creativecommons.org/licenses/by/4.0/
eu_rights_str_mv openAccess
dc.format.none.fl_str_mv application/pdf
dc.publisher.none.fl_str_mv MDPI AG
publisher.none.fl_str_mv MDPI AG
dc.source.none.fl_str_mv reponame:RiuNet. Repositorio Institucional de la Universitat Politécnica de Valéncia
instname:Universitat Politècnica de València (UPV)
instname_str Universitat Politècnica de València (UPV)
reponame_str RiuNet. Repositorio Institucional de la Universitat Politécnica de Valéncia
collection RiuNet. Repositorio Institucional de la Universitat Politécnica de Valéncia
repository.name.fl_str_mv
repository.mail.fl_str_mv
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spelling Personalized Medicine in Infant Population with Cancer: Pharmacogenetic Pilot Study of Polymorphisms Related to Toxicity and Response to ChemotherapyUrtasun, AndreaOlivera, Gladys G.Sendra, LuisAliño, Salvador F.Berlanga, PabloGargallo, PabloBalaguer, JuliaJuan-Ribelles, AntonioAndrés, María del MarCañete, AdelaHerrero, María JoséHervás-Marín, David|||0000-0003-0635-4961PharmacogeneticsSNP (single nucleotide polymorphism)ChemotherapyInfantToxicityTherapeutic efficacyOverall survivalEvent-free survivalAnemiaNeutropeniaThrombocytopeniaESTADISTICA E INVESTIGACION OPERATIVA[EN] Simple Summary Cancer is still the leading cause of disease-related death in pediatric populations and an important source of morbidity. These can be due to the neoplasm itself but also to the treatment administered; infants are patients of special vulnerability. The aim of this work was to identify genetic variants that correlate with significant impacts on treatments' safety and efficacy. 64 oncologic infant patients (under 18 months of age) were genotyped, calling for SNPs (single nucleotide polymorphisms) in genes related to the efficacy and/or toxicity of the chemotherapeutic drugs employed. The relationship of these genetic variants with 37 clinical parameters during 578 chemotherapy cycles was analyzed. Associations were found between 46 SNPs (in genes involved in drug transport and metabolism, gene repair, tumor suppression, and other biological functions) and survival and hematological toxicity. Following studies that confirm these findings, personalized medicine could be offered to improve response and tolerance to chemotherapeutic schemes. Background: Pharmacogenetics is a personalized medicine tool that aims to optimize treatments by adapting them to each individual's genetics, maximizing their efficacy while minimizing their toxicity. Infants with cancer are especially vulnerable, and their co-morbidities have vital repercussions. The study of their pharmacogenetics is new in this clinical field. Methods: A unicentric, ambispective study of a cohort of infants receiving chemotherapy (from January 2007 to August 2019). The genotypes of 64 patients under 18 months of age were correlated with severe drug toxicities and survival. A pharmacogenetics panel was configured based on PharmGKB, drug labels, and international experts' consortiums. Results: Associations between SNPs and hematological toxicity were found. Most meaningful were: MTHFR rs1801131 GT increasing the anemia risk (OR 1.73); rs1517114 GC, XPC rs2228001 GT, increasing neutropenia risk (OR 1.50 and 4.63); ABCB1 rs1045642 AG, TNFRSF11B rs2073618 GG, CYP2B6 rs4802101 TC and SOD2 rs4880 GG increasing thrombocytopenia risk (OR 1.70, 1.77, 1.70, 1.73, respectively). Regarding survival, MTHFR rs1801133 GG, TNFRSF11B rs2073618 GG, XPC rs2228001 GT, CYP3A4 rs2740574 CT, CDA rs3215400 del.del, and SLC01B1 rs4149015 GA were associated with lower overall survival probabilities (HR 3.12, 1.84, 1.68, 2.92, 1.90, and 3.96, respectively). Lastly, for event-free survival, SLC19A1 rs1051266 TT and CDA rs3215400 del.del increased the relapse probability (HR 1.61 and 2.19, respectively). Conclusions: This pharmacogenetic study is a pioneer in dealing with infants under 18 months of age. Further studies are needed to confirm the utility of the findings in this work to be used as predictive genetic biomarkers of toxicity and therapeutic efficacy in the infant population. If confirmed, their use in therapeutic decisions could improve the quality of life and prognosis of these patients.This research was funded by the XIII convocatoria de Ayudas a la Investigación Científica en Salud de la Fundación Mutua Madrileña, Asociación Pablo Ugarte-APU, and Asociación Esperanza y Sonrisa. The L.S. contract is financed by the Infraestructura de Medicina de Precisión asociada a la Ciencia y Tecnología (IMPaCT, IMP/00009). The G.G.O. contract is financed by Asociación Pablo Ugarte-APU.MDPI AGDepartamento de Estadística e Investigación Operativa Aplicadas y CalidadEscuela Politécnica Superior de AlcoyEscuela Técnica Superior de Ingeniería Agronómica y del Medio NaturalAsociación Pablo UgarteInstituto de Salud Carlos IIIRepositorio Institucional de la Universitat Politècnica de València Riunet20232023-03-01journal articlehttp://purl.org/coar/resource_type/c_6501VoRhttp://purl.org/coar/version/c_970fb48d4fbd8a85info:eu-repo/semantics/articleapplication/pdfhttps://riunet.upv.es/handle/10251/203844reponame:RiuNet. Repositorio Institucional de la Universitat Politécnica de Valénciainstname:Universitat Politècnica de València (UPV)InglésengInstituto de Salud Carlos III https://doi.org/10.13039/501100004587 IMP%2F00009open accesshttp://purl.org/coar/access_right/c_abf2Reconocimiento (by)http://creativecommons.org/licenses/by/4.0/info:eu-repo/semantics/openAccessoai:riunet.upv.es:10251/2038442026-06-13T07:49:27Z
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