Antiproliferative effect of natural and semisynthetic polyethers from Laurencia viridis

Squalene-derived polyethers are a unique class of compounds that display a great diversity of structures and a broad array of bioactivities, among which its notable antiproliferative activity stands out against various types of cancer cell lines. In this study, eighteen triterpene squalene-derived p...

Descripción completa

Detalles Bibliográficos
Autores: Santiago-Beníteza, Adrián J., Puerta, Adrián, Padrón, José M., Norte, Manuel, Fernández, José J., Hernández Daranas, Antonio, Cen-Pacheco, Francisco
Tipo de recurso: artículo
Estado:Versión enviada para evaluación y publicación
Fecha de publicación:2024
País:España
Institución:Consejo Superior de Investigaciones Científicas (CSIC)
Repositorio:DIGITAL.CSIC. Repositorio Institucional del CSIC
OAI Identifier:oai:digital.csic.es:10261/345818
Acceso en línea:http://hdl.handle.net/10261/345818
Access Level:acceso abierto
Palabra clave:Squalene-derived triterpenes
Laurencia viridis
Antiproliferative activity
http://metadata.un.org/sdg/15
Protect, restore and promote sustainable use of terrestrial ecosystems, sustainably manage forests, combat desertification, and halt and reverse land degradation and halt biodiversity loss
polyethers
Descripción
Sumario:Squalene-derived polyethers are a unique class of compounds that display a great diversity of structures and a broad array of bioactivities, among which its notable antiproliferative activity stands out against various types of cancer cell lines. In this study, eighteen triterpene squalene-derived polyethers, including twelve natural products and six synthetic derivatives, obtained from the red alga Laurencia viridis Gil-Rodríguez & Haroun were screened for their antiproliferative activity against six cancer cell lines: A549, HBL-100, HeLa, SW1573, T-47D, and WiDr; and a structure-activity relationship (SAR) study was established.