Salvinorin-A induces intense dissociative effects, blocking external sensory perception and modulating interoception and sense of body ownership in humans

Background: Salvinorin-A is a terpene with agonist properties at the kappa-opioid receptor, the binding site of endogenous dynorphins. Salvinorin-A is found in Salvia divinorum, a psychoactive plant traditionally used by the Mazatec people of Oaxaca, Mexico, for medicinal and spiritual purposes. Pre...

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Detalles Bibliográficos
Autores: Maqueda A.E., Valle M., Addy P.H., Antonijoan R.M., Puntes M., Coimbra J., Ballester M.R., Garrido M., González M., Claramunt J., Barker S., Johnson M.W., Griffiths R.R., Riba J.
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2015
País:España
Institución:Institut d’Investigació Biomèdica Sant Pau (IIB Sant Pau)
Repositorio:r-IIB SANT PAU. Repositorio Institucional de Producción Científica del Instituto de Investigación Biomédica Sant Pau
OAI Identifier:oai:iibsantpau.fundanetsuite.com:p10507
Acceso en línea:https://iibsantpau.fundanetsuite.com/Publicaciones/ProdCientif/PublicacionFrw.aspx?id=10507
https://ddd.uab.cat/record/254382
Access Level:acceso abierto
Palabra clave:placebo
salvinorin A
clerodane derivative
psychotropic agent
adult
affect
altered states of consciousness
Article
assessment of humans
body image
cognition
controlled study
double blind procedure
drug effect
female
hallucinogen rating scale
human
interoception
male
multidimensional assessment for interoceptive awareness
normal human
perception
priority journal
sensation
vision
chemically induced
consciousness
dose response
drug effects
hallucination
hearing
organization and management
self concept
verbal communication
young adult
Adult
Auditory Perception
Consciousness
Diterpenes, Clerodane
Dose-Response Relationship, Drug
Double-Blind Method
Female
Hallucinations
Humans
Interoception
Male
Narration
Ownership
Psychotropic Drugs
Self Concept
Visual Perception
Young Adult
Descripción
Sumario:Background: Salvinorin-A is a terpene with agonist properties at the kappa-opioid receptor, the binding site of endogenous dynorphins. Salvinorin-A is found in Salvia divinorum, a psychoactive plant traditionally used by the Mazatec people of Oaxaca, Mexico, for medicinal and spiritual purposes. Previous studies with the plant and salvinorin-A have reported psychedeliclike changes in perception, but also unusual changes in body awareness and detachment from external reality. Here we comprehensively studied the profiles of subjective effects of increasing doses of salvinorin-A in healthy volunteers, with a special emphasis on interoception. Methods: A placebo and three increasing doses of vaporized salvinorin-A (0.25, 0.50, and 1 mg) were administered to eight healthy volunteers with previous experience in the use of psychedelics. Drug effects were assessed using a battery of questionnaires that included, among others, the Hallucinogen Rating Scale, the Altered States of Consciousness, and a new instrument that evaluates different aspects of body awareness: the Multidimensional Assessment for Interoceptive Awareness. Results: Salvinorin-A led to a disconnection from external reality, induced elaborate visions and auditory phenomena, and modified interoception. The lower doses increased somatic sensations, but the highest dose led to a sense of a complete loss of contact with the body. Conclusions: Salvinorin-A induced intense psychotropic effects characterized by a dose-dependent gating of external audiovisual information and an inverted-U dose-response effect on body awareness. These results suggest a prominent role for the kappa opioid receptor in the regulation of sensory perception, interoception, and the sense of body ownership in humans. © The Author 2015.