MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells

Background & Aims: Cholangiocarcinoma (CCA) is a heterogeneous and lethal malignancy, the molecular origins of which remain poorly understood. MicroRNAs (miRs) target diverse signalling pathways, functioning as potent epigenetic regulators of tran-scriptional output. We aimed to characterise miR...

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Autores: Duwe, L. (Lea)|||/items/1df65fa7-63f1-4c57-bb9d-7d33879e5cdb, Munoz-Garrido, P. (Patricia)|||/items/5791e618-3b5a-4fee-935b-e4ef9a792005, Lewinska, M. (Monika)|||/items/1e033557-9622-4746-982f-0fee929aabef, Lafuente-Barquero, J. (Juan)|||/items/b8c028e6-0270-432b-bf89-151996164af3, Satriano, L. (Letizia)|||/items/4dadbe44-845d-4b04-a853-fb105958c197, Hogdall, D. (Dan)|||/items/6081a4f3-817c-46c2-8701-082f39fbe2f4, Taranta, A. (Andrzej)|||/items/23baccb4-878a-41c7-afca-aaae4f253ff0, Nielsen, B.S. (Boye S.)|||/items/5954aa2e-711c-40f5-8fa3-613b29e0d6b8, Ghazal, A. (Awaisa)|||/items/cd460a86-08d7-4735-b982-ab350ffaaeda, Matter, M.S. (Matthias S.)|||/items/47ce053d-852a-4a42-866d-5ddff37ff20b, Banales, J.M. (Jesús M.)|||/items/0c1309ae-e4e4-4e85-b2f1-567a388889d5, Aldana, B.I. (Blanca I.)|||/items/d025dc42-f502-4b2b-8960-428adf46c3ff, Gao, Y.T. (Yu-Tang)|||/items/1309d47b-b519-4f60-96de-558e08f9d0f5, Marquardt, J.U. (Jens U.)|||/items/8893339b-8329-4877-b932-062ad496013c, Roberts, L.R. (Lewis R.)|||/items/53e58801-8eb8-49f9-9fd2-46b93d01e35b, Oliveira, R.C. (Rui C.)|||/items/c1955700-d117-489f-8f07-10e795024300, Koshiol, J. (Jill)|||/items/33448410-bb90-4f8f-89fd-896df187081d, O’Rourke, C.J. (Colm J.)|||/items/087eb514-d64b-470f-92a8-64ed5518c11f, Andersen, J.B. (Jesper B.)|||/items/30522278-e252-4feb-9558-84b5c027103a
Tipo de recurso: artículo
Fecha de publicación:2023
País:España
Institución:Universidad de Navarra
Repositorio:Dadun. Depósito Académico Digital de la Universidad de Navarra
Idioma:inglés
OAI Identifier:oai:dadun.unav.edu:10171/65979
Acceso en línea:https://hdl.handle.net/10171/65979
Access Level:acceso abierto
Palabra clave:Cholangiocarcinoma
Cholangiocytes
FoxO1
microRNAs
Proliferation
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network_name_str España
repository_id_str
spelling MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cellsDuwe, L. (Lea)|||/items/1df65fa7-63f1-4c57-bb9d-7d33879e5cdbMunoz-Garrido, P. (Patricia)|||/items/5791e618-3b5a-4fee-935b-e4ef9a792005Lewinska, M. (Monika)|||/items/1e033557-9622-4746-982f-0fee929aabefLafuente-Barquero, J. (Juan)|||/items/b8c028e6-0270-432b-bf89-151996164af3Satriano, L. (Letizia)|||/items/4dadbe44-845d-4b04-a853-fb105958c197Hogdall, D. (Dan)|||/items/6081a4f3-817c-46c2-8701-082f39fbe2f4Taranta, A. (Andrzej)|||/items/23baccb4-878a-41c7-afca-aaae4f253ff0Nielsen, B.S. (Boye S.)|||/items/5954aa2e-711c-40f5-8fa3-613b29e0d6b8Ghazal, A. (Awaisa)|||/items/cd460a86-08d7-4735-b982-ab350ffaaedaMatter, M.S. (Matthias S.)|||/items/47ce053d-852a-4a42-866d-5ddff37ff20bBanales, J.M. (Jesús M.)|||/items/0c1309ae-e4e4-4e85-b2f1-567a388889d5Aldana, B.I. (Blanca I.)|||/items/d025dc42-f502-4b2b-8960-428adf46c3ffGao, Y.T. (Yu-Tang)|||/items/1309d47b-b519-4f60-96de-558e08f9d0f5Marquardt, J.U. (Jens U.)|||/items/8893339b-8329-4877-b932-062ad496013cRoberts, L.R. (Lewis R.)|||/items/53e58801-8eb8-49f9-9fd2-46b93d01e35bOliveira, R.C. (Rui C.)|||/items/c1955700-d117-489f-8f07-10e795024300Koshiol, J. (Jill)|||/items/33448410-bb90-4f8f-89fd-896df187081dO’Rourke, C.J. (Colm J.)|||/items/087eb514-d64b-470f-92a8-64ed5518c11fAndersen, J.B. (Jesper B.)|||/items/30522278-e252-4feb-9558-84b5c027103aCholangiocarcinomaCholangiocytesFoxO1microRNAsProliferationBackground & Aims: Cholangiocarcinoma (CCA) is a heterogeneous and lethal malignancy, the molecular origins of which remain poorly understood. MicroRNAs (miRs) target diverse signalling pathways, functioning as potent epigenetic regulators of tran-scriptional output. We aimed to characterise miRNome dysregulation in CCA, including its impact on transcriptome homeostasis and cell behaviour.Methods: Small RNA sequencing was performed on 119 resected CCAs, 63 surrounding liver tissues, and 22 normal livers. High -throughput miR mimic screens were performed in three primary human cholangiocyte cultures. Integration of patient tran-scriptomes and miRseq together with miR screening data identified an oncogenic miR for characterization. MiR-mRNA in-teractions were investigated by a luciferase assay. MiR-CRISPR knockout cells were generated and phenotypically characterized in vitro (proliferation, migration, colony, mitochondrial function, glycolysis) and in vivo using subcutaneous xenografts.Results: In total, 13% (140/1,049) of detected miRs were differentially expressed between CCA and surrounding liver tissues, including 135 that were upregulated in tumours. CCA tissues were characterised by higher miRNome heterogeneity and miR biogenesis pathway expression. Unsupervised hierarchical clustering of tumour miRNomes identified three subgroups, including distal CCA-enriched and IDH1 mutant-enriched subgroups. High-throughput screening of miR mimics uncovered 71 miRs that consistently increased proliferation of three primary cholangiocyte models and were upregulated in CCA tissues regardless of anatomical location, among which only miR-27a-3p had consistently increased expression and activity in several cohorts. FoxO signalling was predominantly downregulated by miR-27a-3p in CCA, partially through targeting of FOXO1. MiR-27a knockout increased FOXO1 levels in vitro and in vivo, impeding tumour behaviour and growth.Conclusions: The miRNomes of CCA tissues are highly remodelled, impacting transcriptome homeostasis in part through regulation of transcription factors like FOXO1. MiR-27a-3p arises as an oncogenic vulnerability in CCA.Dadun. Depósito Académico Digital Universidad de Navarra20232023-04-1820232023-01-0120232023-01-01journal articlehttp://purl.org/coar/resource_type/c_6501info:eu-repo/semantics/articleapplication/pdfhttps://hdl.handle.net/10171/65979reponame:Dadun. Depósito Académico Digital de la Universidad de Navarrainstname:Universidad de NavarraInglésengopen accesshttp://purl.org/coar/access_right/c_abf2info:eu-repo/semantics/openAccessoai:dadun.unav.edu:10171/659792026-06-21T12:47:57Z
dc.title.none.fl_str_mv MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells
title MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells
spellingShingle MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells
Duwe, L. (Lea)|||/items/1df65fa7-63f1-4c57-bb9d-7d33879e5cdb
Cholangiocarcinoma
Cholangiocytes
FoxO1
microRNAs
Proliferation
title_short MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells
title_full MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells
title_fullStr MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells
title_full_unstemmed MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells
title_sort MicroRNA-27a-3p targets FoxO signalling to induce tumour-like phenotypes in bile duct cells
dc.creator.none.fl_str_mv Duwe, L. (Lea)|||/items/1df65fa7-63f1-4c57-bb9d-7d33879e5cdb
Munoz-Garrido, P. (Patricia)|||/items/5791e618-3b5a-4fee-935b-e4ef9a792005
Lewinska, M. (Monika)|||/items/1e033557-9622-4746-982f-0fee929aabef
Lafuente-Barquero, J. (Juan)|||/items/b8c028e6-0270-432b-bf89-151996164af3
Satriano, L. (Letizia)|||/items/4dadbe44-845d-4b04-a853-fb105958c197
Hogdall, D. (Dan)|||/items/6081a4f3-817c-46c2-8701-082f39fbe2f4
Taranta, A. (Andrzej)|||/items/23baccb4-878a-41c7-afca-aaae4f253ff0
Nielsen, B.S. (Boye S.)|||/items/5954aa2e-711c-40f5-8fa3-613b29e0d6b8
Ghazal, A. (Awaisa)|||/items/cd460a86-08d7-4735-b982-ab350ffaaeda
Matter, M.S. (Matthias S.)|||/items/47ce053d-852a-4a42-866d-5ddff37ff20b
Banales, J.M. (Jesús M.)|||/items/0c1309ae-e4e4-4e85-b2f1-567a388889d5
Aldana, B.I. (Blanca I.)|||/items/d025dc42-f502-4b2b-8960-428adf46c3ff
Gao, Y.T. (Yu-Tang)|||/items/1309d47b-b519-4f60-96de-558e08f9d0f5
Marquardt, J.U. (Jens U.)|||/items/8893339b-8329-4877-b932-062ad496013c
Roberts, L.R. (Lewis R.)|||/items/53e58801-8eb8-49f9-9fd2-46b93d01e35b
Oliveira, R.C. (Rui C.)|||/items/c1955700-d117-489f-8f07-10e795024300
Koshiol, J. (Jill)|||/items/33448410-bb90-4f8f-89fd-896df187081d
O’Rourke, C.J. (Colm J.)|||/items/087eb514-d64b-470f-92a8-64ed5518c11f
Andersen, J.B. (Jesper B.)|||/items/30522278-e252-4feb-9558-84b5c027103a
author Duwe, L. (Lea)|||/items/1df65fa7-63f1-4c57-bb9d-7d33879e5cdb
author_facet Duwe, L. (Lea)|||/items/1df65fa7-63f1-4c57-bb9d-7d33879e5cdb
Munoz-Garrido, P. (Patricia)|||/items/5791e618-3b5a-4fee-935b-e4ef9a792005
Lewinska, M. (Monika)|||/items/1e033557-9622-4746-982f-0fee929aabef
Lafuente-Barquero, J. (Juan)|||/items/b8c028e6-0270-432b-bf89-151996164af3
Satriano, L. (Letizia)|||/items/4dadbe44-845d-4b04-a853-fb105958c197
Hogdall, D. (Dan)|||/items/6081a4f3-817c-46c2-8701-082f39fbe2f4
Taranta, A. (Andrzej)|||/items/23baccb4-878a-41c7-afca-aaae4f253ff0
Nielsen, B.S. (Boye S.)|||/items/5954aa2e-711c-40f5-8fa3-613b29e0d6b8
Ghazal, A. (Awaisa)|||/items/cd460a86-08d7-4735-b982-ab350ffaaeda
Matter, M.S. (Matthias S.)|||/items/47ce053d-852a-4a42-866d-5ddff37ff20b
Banales, J.M. (Jesús M.)|||/items/0c1309ae-e4e4-4e85-b2f1-567a388889d5
Aldana, B.I. (Blanca I.)|||/items/d025dc42-f502-4b2b-8960-428adf46c3ff
Gao, Y.T. (Yu-Tang)|||/items/1309d47b-b519-4f60-96de-558e08f9d0f5
Marquardt, J.U. (Jens U.)|||/items/8893339b-8329-4877-b932-062ad496013c
Roberts, L.R. (Lewis R.)|||/items/53e58801-8eb8-49f9-9fd2-46b93d01e35b
Oliveira, R.C. (Rui C.)|||/items/c1955700-d117-489f-8f07-10e795024300
Koshiol, J. (Jill)|||/items/33448410-bb90-4f8f-89fd-896df187081d
O’Rourke, C.J. (Colm J.)|||/items/087eb514-d64b-470f-92a8-64ed5518c11f
Andersen, J.B. (Jesper B.)|||/items/30522278-e252-4feb-9558-84b5c027103a
author_role author
author2 Munoz-Garrido, P. (Patricia)|||/items/5791e618-3b5a-4fee-935b-e4ef9a792005
Lewinska, M. (Monika)|||/items/1e033557-9622-4746-982f-0fee929aabef
Lafuente-Barquero, J. (Juan)|||/items/b8c028e6-0270-432b-bf89-151996164af3
Satriano, L. (Letizia)|||/items/4dadbe44-845d-4b04-a853-fb105958c197
Hogdall, D. (Dan)|||/items/6081a4f3-817c-46c2-8701-082f39fbe2f4
Taranta, A. (Andrzej)|||/items/23baccb4-878a-41c7-afca-aaae4f253ff0
Nielsen, B.S. (Boye S.)|||/items/5954aa2e-711c-40f5-8fa3-613b29e0d6b8
Ghazal, A. (Awaisa)|||/items/cd460a86-08d7-4735-b982-ab350ffaaeda
Matter, M.S. (Matthias S.)|||/items/47ce053d-852a-4a42-866d-5ddff37ff20b
Banales, J.M. (Jesús M.)|||/items/0c1309ae-e4e4-4e85-b2f1-567a388889d5
Aldana, B.I. (Blanca I.)|||/items/d025dc42-f502-4b2b-8960-428adf46c3ff
Gao, Y.T. (Yu-Tang)|||/items/1309d47b-b519-4f60-96de-558e08f9d0f5
Marquardt, J.U. (Jens U.)|||/items/8893339b-8329-4877-b932-062ad496013c
Roberts, L.R. (Lewis R.)|||/items/53e58801-8eb8-49f9-9fd2-46b93d01e35b
Oliveira, R.C. (Rui C.)|||/items/c1955700-d117-489f-8f07-10e795024300
Koshiol, J. (Jill)|||/items/33448410-bb90-4f8f-89fd-896df187081d
O’Rourke, C.J. (Colm J.)|||/items/087eb514-d64b-470f-92a8-64ed5518c11f
Andersen, J.B. (Jesper B.)|||/items/30522278-e252-4feb-9558-84b5c027103a
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author
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dc.contributor.none.fl_str_mv Dadun. Depósito Académico Digital Universidad de Navarra
dc.subject.none.fl_str_mv Cholangiocarcinoma
Cholangiocytes
FoxO1
microRNAs
Proliferation
topic Cholangiocarcinoma
Cholangiocytes
FoxO1
microRNAs
Proliferation
description Background & Aims: Cholangiocarcinoma (CCA) is a heterogeneous and lethal malignancy, the molecular origins of which remain poorly understood. MicroRNAs (miRs) target diverse signalling pathways, functioning as potent epigenetic regulators of tran-scriptional output. We aimed to characterise miRNome dysregulation in CCA, including its impact on transcriptome homeostasis and cell behaviour.Methods: Small RNA sequencing was performed on 119 resected CCAs, 63 surrounding liver tissues, and 22 normal livers. High -throughput miR mimic screens were performed in three primary human cholangiocyte cultures. Integration of patient tran-scriptomes and miRseq together with miR screening data identified an oncogenic miR for characterization. MiR-mRNA in-teractions were investigated by a luciferase assay. MiR-CRISPR knockout cells were generated and phenotypically characterized in vitro (proliferation, migration, colony, mitochondrial function, glycolysis) and in vivo using subcutaneous xenografts.Results: In total, 13% (140/1,049) of detected miRs were differentially expressed between CCA and surrounding liver tissues, including 135 that were upregulated in tumours. CCA tissues were characterised by higher miRNome heterogeneity and miR biogenesis pathway expression. Unsupervised hierarchical clustering of tumour miRNomes identified three subgroups, including distal CCA-enriched and IDH1 mutant-enriched subgroups. High-throughput screening of miR mimics uncovered 71 miRs that consistently increased proliferation of three primary cholangiocyte models and were upregulated in CCA tissues regardless of anatomical location, among which only miR-27a-3p had consistently increased expression and activity in several cohorts. FoxO signalling was predominantly downregulated by miR-27a-3p in CCA, partially through targeting of FOXO1. MiR-27a knockout increased FOXO1 levels in vitro and in vivo, impeding tumour behaviour and growth.Conclusions: The miRNomes of CCA tissues are highly remodelled, impacting transcriptome homeostasis in part through regulation of transcription factors like FOXO1. MiR-27a-3p arises as an oncogenic vulnerability in CCA.
publishDate 2023
dc.date.none.fl_str_mv 2023
2023-04-18
2023
2023-01-01
2023
2023-01-01
dc.type.none.fl_str_mv journal article
http://purl.org/coar/resource_type/c_6501
dc.type.openaire.fl_str_mv info:eu-repo/semantics/article
format article
dc.identifier.none.fl_str_mv https://hdl.handle.net/10171/65979
url https://hdl.handle.net/10171/65979
dc.language.none.fl_str_mv Inglés
eng
language_invalid_str_mv Inglés
language eng
dc.rights.none.fl_str_mv open access
http://purl.org/coar/access_right/c_abf2
dc.rights.openaire.fl_str_mv info:eu-repo/semantics/openAccess
rights_invalid_str_mv open access
http://purl.org/coar/access_right/c_abf2
eu_rights_str_mv openAccess
dc.format.none.fl_str_mv application/pdf
dc.source.none.fl_str_mv reponame:Dadun. Depósito Académico Digital de la Universidad de Navarra
instname:Universidad de Navarra
instname_str Universidad de Navarra
reponame_str Dadun. Depósito Académico Digital de la Universidad de Navarra
collection Dadun. Depósito Académico Digital de la Universidad de Navarra
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