Synthesis and stereochemical assignments of diastereomeric Ni(II) complexes of glycine Schiff base with (R)-2-(N-{2-[N-alkyl-N-(1-phenylethyl)-amino]acetyl}amino) benzophenone; a case of configurationally stable stereogenic nitrogen

A family of chiral ligands derived from alpha-phenylethylamine and 2-aminobenzophenone were prepared by alkylation of the nitrogen atom. Upon reaction with glycine and a Ni(II) salt, these ligands were transformed into diastereomeric complexes, as a result of the configurational stability of the ste...

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Detalles Bibliográficos
Autores: Moriwaki, Hiroki, Resch, Daniel, Li, Hengguang, Ojima, Iwao, Takeda, Ryosuke, Aceña Bonilla, José Luis, Soloshonok, Vadym Anatolievch
Tipo de recurso: artículo
Fecha de publicación:2014
País:España
Institución:Universidad del País Vasco
Repositorio:Addi. Archivo Digital para la Docencia y la Investigación
OAI Identifier:oai:addi.ehu.eus:10810/17388
Acceso en línea:http://hdl.handle.net/10810/17388
Access Level:acceso abierto
Palabra clave:amino acids
stereogenic nitrogen
asymmetric synthesis
Ni(II) complexes
Schiff bases
alpha-amino-acids
michael-addition-reactions
substituted pyroglutamic acids
efficient asymmetric-synthesis
phase-transfer catalysts
virtually complete control
alkyl alhide alkylations
large-scale synthesis
nucleophilic glycine
aldol reactions
CHEMISTRY, ORGANIC
Descripción
Sumario:A family of chiral ligands derived from alpha-phenylethylamine and 2-aminobenzophenone were prepared by alkylation of the nitrogen atom. Upon reaction with glycine and a Ni(II) salt, these ligands were transformed into diastereomeric complexes, as a result of the configurational stability of the stereogenic nitrogen atom. Different diastereomeric ratios were observed depending on the substituent R introduced in the starting ligand, and stereochemical assignments were based on X-ray analysis, along with NMR studies and optical rotation measurements.