Curcumin Related 1,4-Diazepines: Regioselective Synthesis, Structure Analysis, Tautomerism, NMR Spectroscopy, X-ray Crystallography, Density Functional Theory and GIAO Calculations

The reaction of 1,2-ethylenediamine with seven fluorinated β-diketones affords two different 1,4-diazepine series depending on the experimental conditions. Their structures as well as tautomerism have been established by 1H, 13C, 15N and 19F nuclear magnetic resonance in solution supported by densit...

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Detalles Bibliográficos
Autores: Andrade, Ana, Torralba, María del Carmen, Torres, M. Rosario, Alkorta, Ibon, Elguero, José, Nieto Gómez, Carla Isabel, Sanz del Castillo, Dionisia, Claramunt, Rosa M.
Tipo de recurso: artículo
Fecha de publicación:2017
País:España
Institución:Universidad Nacional de Educación a Distancia
Repositorio:e-spacio. Repositorio Institucional de la UNED
Idioma:inglés
OAI Identifier:oai:e-spacio.uned.es:20.500.14468/12776
Acceso en línea:https://hdl.handle.net/20.500.14468/12776
Access Level:acceso abierto
Palabra clave:Curcuminoid
Diazepines
Tautomerism
NMR
X-ray
DFT
Descripción
Sumario:The reaction of 1,2-ethylenediamine with seven fluorinated β-diketones affords two different 1,4-diazepine series depending on the experimental conditions. Their structures as well as tautomerism have been established by 1H, 13C, 15N and 19F nuclear magnetic resonance in solution supported by density functional theory calculations at the B3LYP/6-311++G(d,p) level. The two compounds obtained from (E)-5-(2-fluoro-4-hydroxyphenyl)-1-phenylpent-4-ene-1,3-dione were analyzed by X-ray crystallography and studied by solid-state NMR.