Photoswitching endogenous glutamate receptors in neural ensembles and single synapses in vivo

To interrogate animal physiology in vivo, there is a lack of non-genetic methods to control the activity of endogenous proteins with pharmacological and spatiotemporal precision. To address this need, we recently developed targeted covalent photoswitchable (TCP) compounds that enable the remote cont...

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Detalles Bibliográficos
Autores: Garrido-Charles, Aida, Bosch, Miquel, Lee, Hyojung, Rovira, Xavier, Pittolo, Silvia, Llobet, Artur, Wong, Hovy Ho-Wai, Trapero, Ana, Matera, Carlo, Papotto, Claudio, Serra, Carme, Llebaria, Amadeu, Soriano, Eduardo, Sanchez-Vives, Maria V., Holt, Christine E, Gorostiza, Pau
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2025
País:España
Institución:Consejo Superior de Investigaciones Científicas (CSIC)
Repositorio:DIGITAL.CSIC. Repositorio Institucional del CSIC
OAI Identifier:oai:digital.csic.es:10261/399949
Acceso en línea:http://hdl.handle.net/10261/399949
Access Level:acceso abierto
Palabra clave:Pulse-chase
AMPAR
Kainate
Xenopus
Azobenzene
Calcium imaging
Covalent drug
dendritic spines
Hippocampus
Long-term depression
Optopharmacology
Photopharmacology
Photoswitch
Plasticity
Rat
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Descripción
Sumario:To interrogate animal physiology in vivo, there is a lack of non-genetic methods to control the activity of endogenous proteins with pharmacological and spatiotemporal precision. To address this need, we recently developed targeted covalent photoswitchable (TCP) compounds that enable the remote control of endogenous glutamate receptors (GluRs) using light.