Cannabinoid withdrawal syndrome is reduced in pre-proenkephalin knock-out mice

The functional interactions between the endogenous cannabinoid and opioid systems were evaluated in pre-proenkephalin-deficient mice. Antinociception induced in the tail-immersion test by acute Delta9-tetrahydrocannabinol was reduced in mutant mice, whereas no difference between genotypes was observ...

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Detalles Bibliográficos
Autores: Valverde Granados, Olga, Maldonado, Rafael, 1961-, Valjent, Emmanuel, Zimmer, Anne M., Zimmer, Andreas
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2000
País:España
Institución:Universitat Pompeu Fabra
Repositorio:Repositorio Digital de la UPF
OAI Identifier:oai:repositori.upf.edu:10230/16670
Acceso en línea:http://hdl.handle.net/10230/16670
http://dx.doi.org/10.1523/jneurosci.20-24-09284.2000
Access Level:acceso abierto
Palabra clave:Cannabinoides -- Efectes fisiològics
Cannabinoides -- Receptors
Drogoaddicció -- Aspectes moleculars
Cannabinoid
Opioid
Mice
Mutation
Withdrawal
Addiction
Tolerance
Descripción
Sumario:The functional interactions between the endogenous cannabinoid and opioid systems were evaluated in pre-proenkephalin-deficient mice. Antinociception induced in the tail-immersion test by acute Delta9-tetrahydrocannabinol was reduced in mutant mice, whereas no difference between genotypes was observed in the effects induced on body temperature, locomotion, or ring catalepsy. During a chronic treatment with Delta9-tetrahydrocannabinol, the development of tolerance to the analgesic responses induced by this compound was slower in mice lacking enkephalin. In addition, cannabinoid withdrawal syndrome, precipitated in Delta9-tetrahydrocannabinol-dependent mice by the injection of SR141716A, was significantly attenuated in mutant mice. These results indicate that the endogenous enkephalinergic system is involved in the antinociceptive responses of Delta9-tetrahydrocannabinol and participates in the expression of cannabinoid abstinence.