SEAMARK

Patients with both BRAF V600E mutations and microsatellite instability-high (MSI-H)/mismatch repair-deficient (dMMR) metastatic colorectal cancer (mCRC) have poor prognosis. Currently, there are no specifically targeted first-line treatment options indicated for patients with mCRC whose tumors harbo...

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Detalles Bibliográficos
Autores: Elez, Elena|||0000-0002-4653-6324, Kopetz, Scott, Tabernero, Josep|||0000-0002-2495-8139, Bekaii-Saab, Tanios, Taieb, Julien|||0000-0002-9955-4753, Yoshino, Takayuki|||0000-0002-0489-4756, Manji, Gulam, Fernandez, Kathrine, Abbattista, Antonello, Zhang, Xiaosong, Morris, Van K
Tipo de recurso: artículo
Fecha de publicación:2024
País:España
Institución:Universitat Autònoma de Barcelona
Repositorio:Dipòsit Digital de Documents de la UAB
Idioma:inglés
OAI Identifier:oai:ddd.uab.cat:326606
Acceso en línea:https://ddd.uab.cat/record/326606
https://dx.doi.org/urn:doi:10.2217/fon-2022-1249
Access Level:acceso abierto
Palabra clave:BRAF V600
Cetuximab
dMMR
Encorafenib
Immunotherapy
Metastatic colorectal cancer
MSI-H
Pembrolizumab
Targeted therapy
Triplet combination therapy
Descripción
Sumario:Patients with both BRAF V600E mutations and microsatellite instability-high (MSI-H)/mismatch repair-deficient (dMMR) metastatic colorectal cancer (mCRC) have poor prognosis. Currently, there are no specifically targeted first-line treatment options indicated for patients with mCRC whose tumors harbor both molecular aberrations. Pembrolizumab is a checkpoint inhibitor approved for the treatment of MSI-H/dMMR mCRC, and the BRAF inhibitor encorafenib, in combination with cetuximab, is approved for previously treated BRAF V600E-mutant mCRC. Combination of pembrolizumab with encorafenib and cetuximab may synergistically enhance antitumor activity in patients with BRAF V600E-mutant, MSI-H/dMMR mCRC. SEAMARK is a randomized phase II study comparing the efficacy of the combination of pembrolizumab with encorafenib and cetuximab versus pembrolizumab alone in patients with previously untreated BRAF V600E-mutant, MSI-H/dMMR mCRC.