Acquired mechanisms of resistance to osimertinib-the next challenge

EGFR-mutated tumors represent a significant percentage of non-small cell lung cancer. Despite the increasing use of osimertinib, a treatment that has demonstrated an outstanding clinical benefit with a tolerable toxicity profile, EGFR tumors eventually acquire mechanisms of resistance. In the last y...

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Detalles Bibliográficos
Autores: Rios-Hoyo, Alejandro, Moliner Jiménez, Laura, Arriola Aperribay, Edurne
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2022
País:España
Institución:Varias* (Consorci de Biblioteques Universitáries de Catalunya, Centre de Serveis Científics i Acadèmics de Catalunya)
Repositorio:Recercat. Dipósit de la Recerca de Catalunya
OAI Identifier:oai:recercat.cat:10230/54397
Acceso en línea:http://hdl.handle.net/10230/54397
http://dx.doi.org/10.3390/cancers14081931
Access Level:acceso abierto
Palabra clave:EGFR
NSCLC
Mechanisms of resistance
Osimertinib
Descripción
Sumario:EGFR-mutated tumors represent a significant percentage of non-small cell lung cancer. Despite the increasing use of osimertinib, a treatment that has demonstrated an outstanding clinical benefit with a tolerable toxicity profile, EGFR tumors eventually acquire mechanisms of resistance. In the last years, multiple mechanisms of resistance have been identified; however, after progressing on osimertinib, treatment options remain bleak. In this review, we cover the most frequent alterations and potential therapeutic strategies to overcome them.