FDA-approved antivirals ledipasvir and daclatasvir downregulate the Src-EPHA2-Akt oncogenic pathway in colorectal and triple-negative breast cancer cells

SRC transformed SW620 cells were a kind gift from Serge Roche (CNRS and University of Montpellier). TRIB2 plasmids were a kind gift from Patrick Eyers (University of Liverpool) and the protein was produced and purified by Andras Lang. This work was funded by grants from the Generalitat de Catalunya...

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Detalles Bibliográficos
Autores: Mezquita, Betlem, Reyes-Farias, Marjorie, Pons, Miquel
Tipo de recurso: artículo
Fecha de publicación:2024
País:España
Institución:Varias* (Consorci de Biblioteques Universitáries de Catalunya, Centre de Serveis Científics i Acadèmics de Catalunya)
Repositorio:Recercat. Dipósit de la Recerca de Catalunya
OAI Identifier:oai:recercat.cat:20.500.12328/4488
Acceso en línea:http://hdl.handle.net/20.500.12328/4488
https://dx.doi.org/10.1016/j.biopha.2024.117325
Access Level:acceso abierto
Palabra clave:Reutilització de fàrmacs
Antivirals d'acció directa
Orientació Src en tumors sòlids
Akt
Proteïna receptora de cèl·lules epitelials tirosina
Quinasa
Receptor d'efrina tipus A 2
ECK
Receptor EPH A2
Proteïna quinasa B
Reutilización de fármacos
Antivirales de acción directa
Orientación a Src en tumores sólidos
Receptor de células epiteliales de la proteína tirosina quinasa
Receptor efrina tipo A 2
Proteína quinasa B
Drug repurposing
Direct-acting antivirals
Src targeting in solid tumors
Epithelial Cell Receptor Protein Tyrosine
Kinase
Ephrin type-A receptor 2
EPH receptor A2
Protein kinase B
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Descripción
Sumario:SRC transformed SW620 cells were a kind gift from Serge Roche (CNRS and University of Montpellier). TRIB2 plasmids were a kind gift from Patrick Eyers (University of Liverpool) and the protein was produced and purified by Andras Lang. This work was funded by grants from the Generalitat de Catalunya (2021 SGR 425) and the Spanish “Agencia Estatal de Investigacion´ ”: PDC2021–121629-I00 (with the support of the Recovery and Resilience Mechanism and NextGenerationEU funding); PID2019–104914RB-I00, and PID2022–139160OB-I00 (with a contribution from European Regional Development funds).