Direct and specific inhibition of factor Xa: an emerging therapeutic strategy for atherothrombotic disease

Atherosclerotic disease is the leading cause of morbidity and mortality worldwide. Despite advances in the medical treatment to acute coronary syndrome (ACS), the mortality and recurrence of ACS are still exceedingly high, thus further treatment optimization is needed. The need to reduce future card...

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Detalles Bibliográficos
Autores: Santos-Gallego, CG, Badimon, L, Badimon, JJ
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2014
País:España
Institución:Institut d’Investigació Biomèdica Sant Pau (IIB Sant Pau)
Repositorio:r-IIB SANT PAU. Repositorio Institucional de Producción Científica del Instituto de Investigación Biomédica Sant Pau
OAI Identifier:oai:iibsantpau.fundanetsuite.com:p9465
Acceso en línea:https://iibsantpau.fundanetsuite.com/Publicaciones/ProdCientif/PublicacionFrw.aspx?id=9465
Access Level:acceso abierto
Palabra clave:Acute coronary syndrome
Myocardial infarction
Anticoagulants
Vitamin K inhibitors
Coagulation
Factor X
Xa inhibitors
Secondary prevention
Descripción
Sumario:Atherosclerotic disease is the leading cause of morbidity and mortality worldwide. Despite advances in the medical treatment to acute coronary syndrome (ACS), the mortality and recurrence of ACS are still exceedingly high, thus further treatment optimization is needed. The need to reduce future cardiovascular events has led to the development of novel therapies to prevent coronary thrombosis, targeting the coagulation pathway, specifically active factor X (Xa). Several factor Xa inhibitors (rivaroxaban, apixaban, darexaban, otamixaban) have been recently developed and studied in the context of ACS. This article critically reviews the comparative mechanisms of action, the risks and benefits, together with the clinical evidence base for the use of these novel Xa inhibitors in the management of ACS patients.