Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation

Alzheimer's disease (AD) is characterised by the presence of extracellular amyloid plaques in the brain. They are composed of aggregated amyloid beta-peptide (Aβ) misfolded into beta-sheets which are the cause of the AD memory impairment and dementia. Memory depends on the hippocampal forma...

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Autores: Picón-Pagès, Pol, Fanlo-Ucar, Hugo, Herrera-Fernández, Víctor, Ausellé Bosch, Sira, Galera López, Lorena, 1993-, Gutiérrez, Daniela A., Ozaita Mintegui, Andrés, 1969-, Álvarez, Alejandra R., Oliva Miguel, Baldomero, Muñoz López, Francisco José, 1964-
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2022
País:España
Institución:Universitat Pompeu Fabra
Repositorio:Repositorio Digital de la UPF
OAI Identifier:oai:repositori.upf.edu:10230/55312
Acceso en línea:http://hdl.handle.net/10230/55312
http://dx.doi.org/10.3390/ijms232315169
Access Level:acceso abierto
Palabra clave:Alzheimer’s disease
CREB
CaMKIIα
Amyloid
Oxidative stress
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spelling Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidationPicón-Pagès, PolFanlo-Ucar, HugoHerrera-Fernández, VíctorAusellé Bosch, SiraGalera López, Lorena, 1993-Gutiérrez, Daniela A.Ozaita Mintegui, Andrés, 1969-Álvarez, Alejandra R.Oliva Miguel, BaldomeroMuñoz López, Francisco José, 1964-Alzheimer’s diseaseCREBCaMKIIαAmyloidOxidative stressAlzheimer's disease (AD) is characterised by the presence of extracellular amyloid plaques in the brain. They are composed of aggregated amyloid beta-peptide (Aβ) misfolded into beta-sheets which are the cause of the AD memory impairment and dementia. Memory depends on the hippocampal formation and maintenance of synapses by long-term potentiation (LTP), whose main steps are the activation of NMDA receptors, the phosphorylation of CaMKIIα and the nuclear translocation of the transcription factor CREB. It is known that Aβ oligomers (oAβ) induce synaptic loss and impair the formation of new synapses. Here, we have studied the effects of oAβ on CaMKIIα. We found that oAβ produce reactive oxygen species (ROS), that induce CaMKIIα oxidation in human neuroblastoma cells as we assayed by western blot and immunofluorescence. Moreover, this oxidized isoform is significantly present in brain samples from AD patients. We found that the oxidized CaMKIIα is active independently of the binding to calcium/calmodulin, and that CaMKIIα phosphorylation is mutually exclusive with CaMKIIα oxidation as revealed by immunoprecipitation and western blot. An in silico modelling of the enzyme was also performed to demonstrate that oxidation induces an activated state of CaMKIIα. In brains from AD transgenic models of mice and in primary cultures of murine hippocampal neurons, we demonstrated that the oxidation of CaMKIIα induces the phosphorylation of CREB and its translocation to the nucleus to promote the transcription of ARC and BDNF. Our data suggests that CaMKIIα oxidation would be a pro-survival mechanism that is triggered when a noxious stimulus challenges neurons as do oAβ.This work was supported by the Spanish Ministry of Science and Innovation and Agencia Estatal de Investigación plus FEDER Funds through grants PID2020-117691RB-I00/AEI/10.13039/501100011033 (F.J.M.), SAF2017-83372-R (F.J.M.), BIO 2020-113203RB (B.O.) and PID2021-123482OB-I00 (A.O.). This work was also funded by the “María de Maetzu Programme” for Units of Excellence in R&D and the MM-MELIS intercollaborative projects (award CEX2018-000792-M/IPEP-MM2020-5). Funding for this project was also from the Comisión Nacional de Investigación Científica y Tecnológica-Chile: Fondecyt 12011668 (to A.R.Á.) and Millennium Science Initiative Program—ICN09_016/ICN 2021_045 (to A.R.Á.).MDPI202320232022info:eu-repo/semantics/articleinfo:eu-repo/semantics/publishedVersionapplication/pdfapplication/pdfhttp://hdl.handle.net/10230/55312http://dx.doi.org/10.3390/ijms232315169reponame:Repositorio Digital de la UPFinstname:Universitat Pompeu FabraInglésInt J Mol Sci. 2022 Dec 2;23(23):15169info:eu-repo/grantAgreement/ES/2PE/PID2020-117691RB-I00info:eu-repo/grantAgreement/ES/2PE/SAF2017-83372-Rinfo:eu-repo/grantAgreement/ES/1PE/BIO2020-113203RBinfo:eu-repo/grantAgreement/ES/2PE/PID2021-123482OB-I00© 2022 by the authors. Licensee MDPI, Basel, Switzerland. This article is an open access article distributed under the terms and conditions of the Creative Commons Attribution (CC BY) license (https://creativecommons.org/licenses/by/4.0/).https://creativecommons.org/licenses/by/4.0/info:eu-repo/semantics/openAccessoai:repositori.upf.edu:10230/553122026-06-12T07:21:37Z
dc.title.none.fl_str_mv Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation
title Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation
spellingShingle Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation
Picón-Pagès, Pol
Alzheimer’s disease
CREB
CaMKIIα
Amyloid
Oxidative stress
title_short Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation
title_full Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation
title_fullStr Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation
title_full_unstemmed Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation
title_sort Amyloid β-peptide causes the permanent activation of CaMKIIα through its oxidation
dc.creator.none.fl_str_mv Picón-Pagès, Pol
Fanlo-Ucar, Hugo
Herrera-Fernández, Víctor
Ausellé Bosch, Sira
Galera López, Lorena, 1993-
Gutiérrez, Daniela A.
Ozaita Mintegui, Andrés, 1969-
Álvarez, Alejandra R.
Oliva Miguel, Baldomero
Muñoz López, Francisco José, 1964-
author Picón-Pagès, Pol
author_facet Picón-Pagès, Pol
Fanlo-Ucar, Hugo
Herrera-Fernández, Víctor
Ausellé Bosch, Sira
Galera López, Lorena, 1993-
Gutiérrez, Daniela A.
Ozaita Mintegui, Andrés, 1969-
Álvarez, Alejandra R.
Oliva Miguel, Baldomero
Muñoz López, Francisco José, 1964-
author_role author
author2 Fanlo-Ucar, Hugo
Herrera-Fernández, Víctor
Ausellé Bosch, Sira
Galera López, Lorena, 1993-
Gutiérrez, Daniela A.
Ozaita Mintegui, Andrés, 1969-
Álvarez, Alejandra R.
Oliva Miguel, Baldomero
Muñoz López, Francisco José, 1964-
author2_role author
author
author
author
author
author
author
author
author
dc.subject.none.fl_str_mv Alzheimer’s disease
CREB
CaMKIIα
Amyloid
Oxidative stress
topic Alzheimer’s disease
CREB
CaMKIIα
Amyloid
Oxidative stress
description Alzheimer's disease (AD) is characterised by the presence of extracellular amyloid plaques in the brain. They are composed of aggregated amyloid beta-peptide (Aβ) misfolded into beta-sheets which are the cause of the AD memory impairment and dementia. Memory depends on the hippocampal formation and maintenance of synapses by long-term potentiation (LTP), whose main steps are the activation of NMDA receptors, the phosphorylation of CaMKIIα and the nuclear translocation of the transcription factor CREB. It is known that Aβ oligomers (oAβ) induce synaptic loss and impair the formation of new synapses. Here, we have studied the effects of oAβ on CaMKIIα. We found that oAβ produce reactive oxygen species (ROS), that induce CaMKIIα oxidation in human neuroblastoma cells as we assayed by western blot and immunofluorescence. Moreover, this oxidized isoform is significantly present in brain samples from AD patients. We found that the oxidized CaMKIIα is active independently of the binding to calcium/calmodulin, and that CaMKIIα phosphorylation is mutually exclusive with CaMKIIα oxidation as revealed by immunoprecipitation and western blot. An in silico modelling of the enzyme was also performed to demonstrate that oxidation induces an activated state of CaMKIIα. In brains from AD transgenic models of mice and in primary cultures of murine hippocampal neurons, we demonstrated that the oxidation of CaMKIIα induces the phosphorylation of CREB and its translocation to the nucleus to promote the transcription of ARC and BDNF. Our data suggests that CaMKIIα oxidation would be a pro-survival mechanism that is triggered when a noxious stimulus challenges neurons as do oAβ.
publishDate 2022
dc.date.none.fl_str_mv 2022
2023
2023
dc.type.none.fl_str_mv info:eu-repo/semantics/article
info:eu-repo/semantics/publishedVersion
format article
status_str publishedVersion
dc.identifier.none.fl_str_mv http://hdl.handle.net/10230/55312
http://dx.doi.org/10.3390/ijms232315169
url http://hdl.handle.net/10230/55312
http://dx.doi.org/10.3390/ijms232315169
dc.language.none.fl_str_mv Inglés
language_invalid_str_mv Inglés
dc.relation.none.fl_str_mv Int J Mol Sci. 2022 Dec 2;23(23):15169
info:eu-repo/grantAgreement/ES/2PE/PID2020-117691RB-I00
info:eu-repo/grantAgreement/ES/2PE/SAF2017-83372-R
info:eu-repo/grantAgreement/ES/1PE/BIO2020-113203RB
info:eu-repo/grantAgreement/ES/2PE/PID2021-123482OB-I00
dc.rights.none.fl_str_mv https://creativecommons.org/licenses/by/4.0/
info:eu-repo/semantics/openAccess
rights_invalid_str_mv https://creativecommons.org/licenses/by/4.0/
eu_rights_str_mv openAccess
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dc.publisher.none.fl_str_mv MDPI
publisher.none.fl_str_mv MDPI
dc.source.none.fl_str_mv reponame:Repositorio Digital de la UPF
instname:Universitat Pompeu Fabra
instname_str Universitat Pompeu Fabra
reponame_str Repositorio Digital de la UPF
collection Repositorio Digital de la UPF
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