Structural study of 3-methyl-3-azabicyclo[3.2.1]octan-8α(and β)-ols by ab initio calculations, NMR and IR spectroscopy

A stereoselective synthesis of 3-methyl-3-azabicyclo[3.2.1]octan-8α(and β)-ols (I and II) has been carried out. Compounds I and II have been studied by 1H, 13C NMR, NOE 1D experiments, IR spectroscopy and ab initio calculations. These compounds (I and II) adopt in CDCl3 a preferred chair-envelope co...

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Detalles Bibliográficos
Autores: Iriepa, Isabel, Madrid, A. I., Morreale, Antonio, Gálvez-Ruano, Enrique, Bellanato, Juana
Tipo de recurso: artículo
Estado:Versión aceptada para publicación
Fecha de publicación:2003
País:España
Institución:Consejo Superior de Investigaciones Científicas (CSIC)
Repositorio:DIGITAL.CSIC. Repositorio Institucional del CSIC
OAI Identifier:oai:digital.csic.es:10261/243720
Acceso en línea:http://hdl.handle.net/10261/243720
Access Level:acceso abierto
Palabra clave:3-methyl-3-azabicyclo[3.2.1]octan-8α(and β)-ols
Infrared spectroscopy
NMR spectroscopy
Conformational analysis
Ab initio calculations
Descripción
Sumario:A stereoselective synthesis of 3-methyl-3-azabicyclo[3.2.1]octan-8α(and β)-ols (I and II) has been carried out. Compounds I and II have been studied by 1H, 13C NMR, NOE 1D experiments, IR spectroscopy and ab initio calculations. These compounds (I and II) adopt in CDCl3 a preferred chair-envelope conformation with the N–CH3 group in equatorial position. Intermolecular associations were deduced by IR and ab initio calculations. The infrared spectra in the ν(O–H) region of compounds I and II were compared with the spectra theoretically calculated at the B3LYP/6-311G** level. Good agreement between the experimental observations and the theoretical calculations has been found.