Vortioxetine in major depressive disorder

Introduction: Vortioxetine is a multimodal-acting antidepressant that provides improvements on cognitive function aside from antidepressants and anxiolytic effects. Vortioxetine has been found to be one of the most effective and best tolerated options for major depressive disorder (MDD) in head-to-h...

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Detalles Bibliográficos
Autores: Diego-Adeliño, Javier de|||0000-0001-9708-2441, Crespo, José Manuel, Mora, Fernando|||0000-0003-4698-1679, Neyra, Adrián, Iborra, Pedro|||0000-0001-9041-0983, Gutiérrez-Rojas, Luis|||0000-0003-0082-2189, Salonia, Selman F.
Tipo de recurso: artículo
Fecha de publicación:2022
País:España
Institución:Universitat Autònoma de Barcelona
Repositorio:Dipòsit Digital de Documents de la UAB
Idioma:inglés
OAI Identifier:oai:ddd.uab.cat:277681
Acceso en línea:https://ddd.uab.cat/record/277681
https://dx.doi.org/urn:doi:10.1080/14740338.2022.2019705
Access Level:acceso abierto
Palabra clave:Antidepressant
Cognition
Efficacy
Interactions
Major depressive disorder
Neurotransmission
Pharmacology
Safety
Vortioxetine
Descripción
Sumario:Introduction: Vortioxetine is a multimodal-acting antidepressant that provides improvements on cognitive function aside from antidepressants and anxiolytic effects. Vortioxetine has been found to be one of the most effective and best tolerated options for major depressive disorder (MDD) in head-to-head trials. Areas covered: The present review intends to gather the most relevant and pragmatic data of vortioxetine in MDD, specially focusing on new studies that emerged between 2015 and 2020. Expert opinion: Vortioxetine is the first antidepressant that has shown improvements both in depression and cognitive symptoms, due to the unique multimodal mechanism of action that combine the 5-HT reuptake inhibition with modulations of other key pre- and post-synaptic 5-HT receptors (agonism of 5-HT receptor, partial agonism of 5-HT receptor, and antagonism of 5-HT, 5-HT and 5-HT receptors). This new mechanism of action can explain the dose-dependent effect and can be responsible for its effects on cognitive functioning and improved tolerability profile. Potential analgesic and anti-inflammatory properties observed in preclinical studies as well as interesting efficacy and tolerability results of clinical studies with specific target groups render it a promising therapeutic option for patients with MDD and concomitant conditions (as menopause symptoms, pain, inflammation, apathy, sleep and/or metabolic abnormalities).