Diazo group as a new chemical reporter for bioorthogonal labelling of biomolecules

Diazoacetyl groups have been shown to undergo spontaneous cycloaddition reactions with strained alkenes and alkynes. The rates of reaction are similar to the equivalent reactions of azide groups. This allows diazo groups to be used as bioorthogonal reporter groups. This is demonstrated by fluorescen...

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Detalles Bibliográficos
Autores: Josa-Culleré, Laia, Wainman, Yelena A., Brindle, Kevin M., Leeper, Finian J.
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2014
País:España
Institución:Consejo Superior de Investigaciones Científicas (CSIC)
Repositorio:DIGITAL.CSIC. Repositorio Institucional del CSIC
OAI Identifier:oai:digital.csic.es:10261/413052
Acceso en línea:http://hdl.handle.net/10261/413052
https://api.elsevier.com/content/abstract/scopus_id/84908228871
Access Level:acceso abierto
Palabra clave:Diazoacetyl groups
Medicinal chemistry
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Descripción
Sumario:Diazoacetyl groups have been shown to undergo spontaneous cycloaddition reactions with strained alkenes and alkynes. The rates of reaction are similar to the equivalent reactions of azide groups. This allows diazo groups to be used as bioorthogonal reporter groups. This is demonstrated by fluorescent labelling of a diazoacetylated protein and of cell-surface glycans via metabolic incorporation of a diazoacetylated sugar. This journal is