Extended hildebrand solubility approach applied to nimodipine in peg 400 + ethanol mixtures

Nimodipine (NMD) is a drug used as cerebral vasodilator whose physicochemical properties in solution have not been studied completely. In this work the Extended Hildebrand Solubility Approach (EHSA) was applied to evaluate the equilibrium solubility of NMD in some polyethylene glycol 400 + ethanol m...

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Detalles Bibliográficos
Autores: Gómez, Jorge L., Rodríguez, Gerson A., Cristancho, Diana M., Delgado, Daniel R., Mora, Carolina P., Yurquina, Alicia, Martínez, Fleming
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2013
País:Colombia
Institución:Universidad Nacional de Colombia
Repositorio:Repositorio UN
Idioma:español
OAI Identifier:oai:repositorio.unal.edu.co:unal/49322
Acceso en línea:https://repositorio.unal.edu.co/handle/unal/49322
http://bdigital.unal.edu.co/42779/
http://bdigital.unal.edu.co/42779/2/
Access Level:acceso abierto
Palabra clave:nimodipina
PEG 400 + etanol
Método Extendido de Solubilidad de Hildebrand
mezclas binarias
parámetro de solubilidad
Nimodipine
PEG 400 + ethanol
Extended Hildebrand Solubility Approach
binary mixtures
solubility parameter
Descripción
Sumario:Nimodipine (NMD) is a drug used as cerebral vasodilator whose physicochemical properties in solution have not been studied completely. In this work the Extended Hildebrand Solubility Approach (EHSA) was applied to evaluate the equilibrium solubility of NMD in some polyethylene glycol 400 + ethanol mixtures at 298.15 K. An acceptable correlative capacity of EHSA was found using a regular polynomial model in order three (overall deviation lower than 1.3%), when the W interaction parameter is related to the solubility parameter of the mixtures. Moreover, the mean deviation obtained in the estimated solubility with respect to experimental solubility was lower than the one obtained directly by means of an empiric regression in order three of the logarithm experimental solubility as a function of the mixtures' solubility parameters (1.7%).