HA1077 inhibits cell proliferation of oral squamous cell carcinoma in vitro

Oral squamous cell carcinoma is a common malignant lesion. ROCKs proteins are associated with pathogenesis and progression of human tumours. This study aimed to evaluate the functional role of ROCKs in the regulation of cell proliferation of oral squamous cell carcinoma in vitro. BrdU incorporation...

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Detalles Bibliográficos
Autores: Borges, Guilherme Henrique, Carboni, Simone de Sales Costa Moreira, Carneiro, Anna Cecília Dias Maciel, Hiss, Lorraine Stephanie, Silveira, Isadora Caixeta da, Crema, Virginia Oliveira
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2022
País:Brasil
Institución:Universidade Federal de Itajubá (UNIFEI)
Repositorio:Research, Society and Development
Idioma:inglés
OAI Identifier:oai:ojs.pkp.sfu.ca:article/26730
Acceso en línea:https://rsdjournal.org/index.php/rsd/article/view/26730
Access Level:acceso abierto
Palabra clave:Cell proliferation
HA-1077
Oral squamous cell carcinoma
ROCKs
SCC-4
Y-27632.
Proliferação celular
Carcinoma de células escamosas oral
Proliferación celular
Carcinoma oral de células escamosas
Descripción
Sumario:Oral squamous cell carcinoma is a common malignant lesion. ROCKs proteins are associated with pathogenesis and progression of human tumours. This study aimed to evaluate the functional role of ROCKs in the regulation of cell proliferation of oral squamous cell carcinoma in vitro. BrdU incorporation assays and KI-67 immunoexpression were performed by using SCC-4 cell line from oral squamous cell carcinoma. Control and treated cells: HA-1077 (25, 50 and 100 μmol/l), 50 μmol HA-1077 and Y-27632 30 μmol/l, Y-27632 30 μmol/l were cutured for 6 h. The number of SCC-4 cells treated with: HA-1077 (25, 50 and 100 μmol/l), HA-1077 50 μmol/l and/or Y-27632 30 μmol/l was significantly lower than control cells in BrdU assay [F (5.17) = 443.818, p<0.0001] and in KI-67 assay [F = 192.595, d.f. = 5,17; p<0.0001]. The results obtained suggest that the pathways that evolve ROCKs proteins play an important functional role in the positive regulation of cell proliferation in oral squamous cell carcinoma.