Zoledronate and related impurities analysis by capillary zone electrophoresis

A capillary zone electrophoretic (CZE) method has been developed for the determination of zoledronate and its related impurities (phosphyte and phosphate). Successful separation of the drug from the impurities was achieved using 7.5 mM of phthalic acid adjusted to pH 3.50 with TRIS, as background el...

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Detalles Bibliográficos
Autores: Alvarez, Gisela Solange, Foglia, María Lucía, Camporotondi, Daniela Edhit, Giorgieri, Sergio, Desimone, Martín Federico, Diaz, Luis Eduardo
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2014
País:Argentina
Institución:Consejo Nacional de Investigaciones Científicas y Técnicas
Repositorio:CONICET Digital (CONICET)
Idioma:inglés
OAI Identifier:oai:ri.conicet.gov.ar:11336/30729
Acceso en línea:http://hdl.handle.net/11336/30729
Access Level:acceso abierto
Palabra clave:Capillary Zone Electrophoresis
Zoledronate
Biphosphonates
Impurities
https://purl.org/becyt/ford/1.4
https://purl.org/becyt/ford/1
Descripción
Sumario:A capillary zone electrophoretic (CZE) method has been developed for the determination of zoledronate and its related impurities (phosphyte and phosphate). Successful separation of the drug from the impurities was achieved using 7.5 mM of phthalic acid adjusted to pH 3.50 with TRIS, as background electrolyte with an indirect detection at 205 nm. The optimized method was validated for specificity, precision, linearity and accuracy. The limit of detection was 1.8 µg ml-1 and the limit of quantification was 5.9 µg ml-1 for phosphyte. The limit of detection was 2.8 µg ml-1 and the limit of quantification was 9.3 µg ml-1 for phosphate. The developed CZE method used to determine zoledronate, phosphyte and phosphate as bisphosphonates impurities can be used to evaluate the quality of regular production samples of zoledronate.