Cyclodextrin complexes for treatment improvement in infectious diseases

Infectious diseases are a heterogeneous group of maladies that represent a serious burden to healthcare systems worldwide. Most of the available antimicrobial drugs display poor biopharmaceutical properties that compromise their effectiveness. Cyclodextrins (CDs) are cyclic oligosaccharides of gluco...

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Detalhes bibliográficos
Autores: Imperiale, Julieta Celeste, Sosnik, Alejandro Dario
Tipo de documento: artigo
Estado:Versão publicada
Data de publicação:2015
País:Argentina
Recursos:Consejo Nacional de Investigaciones Científicas y Técnicas
Repositório:CONICET Digital (CONICET)
Idioma:inglês
OAI Identifier:oai:ri.conicet.gov.ar:11336/84671
Acesso em linha:http://hdl.handle.net/11336/84671
Access Level:Acceso aberto
Palavra-chave:CYCLODEXTRINS
DRUG/CYCLODEXTRIN COMPLEX
INFECTIOUS DISEASES
LOW PHYSICAL STABILITY
POOR AQUEOUS SOLUBILITY
https://purl.org/becyt/ford/2.10
https://purl.org/becyt/ford/2
Descrição
Resumo:Infectious diseases are a heterogeneous group of maladies that represent a serious burden to healthcare systems worldwide. Most of the available antimicrobial drugs display poor biopharmaceutical properties that compromise their effectiveness. Cyclodextrins (CDs) are cyclic oligosaccharides of glucopyranose formed by a variable number of repeating units that combine a hydrophilic surface with a hydrophobic cavity. The production of drug/CD complexes has become one of the most extensively investigated technology approaches to improve the stability, solubility, dissolution rate and bioavailability of drugs. The present work overviews the applications of CDs for the formulation of anti-infective agents along with the most relevant administration routes. Finally, an update on the complexes with CDs available on the market to treat infectious diseases is presented.