Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s

Cystic echinococcosis is a zoonotic disease caused by the parasite Echinococcus granulosus sensu lato (s.l.), which is worldwide distributed and causes long-lasting infections in animals and humans. The existing treatment is limited to the use of benzimidazoles, mainly albendazole (ABZ). However, it...

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Autores: Albani, Clara Maria, Borgo, Jimena, Fabbri, Julia, Pensel, Patricia Eugenia, Fasciani, L., Elso, Orlando German, Papademetrio, Daniela Laura, Grasso, Daniel Hector, Paladini, A., Beer, Maria Florencia, Farias, Nahuel Emiliano, Elissondo, N., Gambino, G., Zoppi, J., Sülsen, Valeria Patricia, Elissondo, María Celina
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2022
País:Argentina
Institución:Consejo Nacional de Investigaciones Científicas y Técnicas
Repositorio:CONICET Digital (CONICET)
Idioma:inglés
OAI Identifier:oai:ri.conicet.gov.ar:11336/211604
Acceso en línea:http://hdl.handle.net/11336/211604
Access Level:acceso abierto
Palabra clave:Asteraceae
Echinococcus granulosus
Cystic echinococcosis
https://purl.org/becyt/ford/3.3
https://purl.org/becyt/ford/3
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network_acronym_str AR
network_name_str Argentina
repository_id_str
dc.title.none.fl_str_mv Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s
title Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s
spellingShingle Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s
Albani, Clara Maria
Asteraceae
Echinococcus granulosus
Cystic echinococcosis
https://purl.org/becyt/ford/3.3
https://purl.org/becyt/ford/3
title_short Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s
title_full Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s
title_fullStr Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s
title_full_unstemmed Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s
title_sort Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s
dc.creator.none.fl_str_mv Albani, Clara Maria
Borgo, Jimena
Fabbri, Julia
Pensel, Patricia Eugenia
Fasciani, L.
Elso, Orlando German
Papademetrio, Daniela Laura
Grasso, Daniel Hector
Paladini, A.
Beer, Maria Florencia
Farias, Nahuel Emiliano
Elissondo, N.
Gambino, G.
Zoppi, J.
Sülsen, Valeria Patricia
Elissondo, María Celina
author Albani, Clara Maria
author_facet Albani, Clara Maria
Borgo, Jimena
Fabbri, Julia
Pensel, Patricia Eugenia
Fasciani, L.
Elso, Orlando German
Papademetrio, Daniela Laura
Grasso, Daniel Hector
Paladini, A.
Beer, Maria Florencia
Farias, Nahuel Emiliano
Elissondo, N.
Gambino, G.
Zoppi, J.
Sülsen, Valeria Patricia
Elissondo, María Celina
author_role author
author2 Borgo, Jimena
Fabbri, Julia
Pensel, Patricia Eugenia
Fasciani, L.
Elso, Orlando German
Papademetrio, Daniela Laura
Grasso, Daniel Hector
Paladini, A.
Beer, Maria Florencia
Farias, Nahuel Emiliano
Elissondo, N.
Gambino, G.
Zoppi, J.
Sülsen, Valeria Patricia
Elissondo, María Celina
author2_role author
author
author
author
author
author
author
author
author
author
author
author
author
author
author
dc.subject.none.fl_str_mv Asteraceae
Echinococcus granulosus
Cystic echinococcosis
https://purl.org/becyt/ford/3.3
https://purl.org/becyt/ford/3
topic Asteraceae
Echinococcus granulosus
Cystic echinococcosis
https://purl.org/becyt/ford/3.3
https://purl.org/becyt/ford/3
description Cystic echinococcosis is a zoonotic disease caused by the parasite Echinococcus granulosus sensu lato (s.l.), which is worldwide distributed and causes long-lasting infections in animals and humans. The existing treatment is limited to the use of benzimidazoles, mainly albendazole (ABZ). However, it has unwanted side effects and its efficacy is about 50%. The Asteraceae family includes plants that have therapeutic applications (medicinal species) and has an important role in new drug development. The species belonging to a different genus of this family show a wide range of anti-inflammatory, antimicrobial, antioxidant, hepatoprotective, and antiparasitic activities, among others. The aim of the present study was to evaluate the in vitro efficacy of extracts of four Asteraceae species against protoscoleces of E. granulosus sensu stricto (s.s.). On the other hand, the Stevia aristata extract was assessed on the murine cyst of E. granulosus (s.s.) and the efficacy of S. aristata extract was investigated in a murine model of CE. Stevia satureiifolia, S. aristata, Grindelia pulchella, and G. chiloensis extracts at 100 μg/mL caused a decrease in protoscoleces viability; however, S. aristata extract produced the greatest in vitro protoscolicidal effect. After 20 days of treatment with the highest concentration (100 μg/mL) of S. aristata extract, protoscoleces viability decreased to 0%. The tegumental changes observed by scanning electron microscopy were consistent with the reduction in vitality. The collapse of the germinal layer was registered in 60 ± 5.8% and 83.3 ± 12.0% of cysts treated during 4 days with 50 and 100 μg/ml, respectively. The half maximal effective concentration (EC50) value of the S. aristata extract against E. granulosus (s.s.) cysts was 47.86 μg/mL (96 h). The dosage of infected animals with the 50 mg kg-1 dose of S. aristata extract resulted in a significant reduction in cyst weight in comparison with the control group. In conclusion, S. aristata extract was demonstrated to exert a marked effect, both in vitro and in the murine model.
publishDate 2022
dc.date.none.fl_str_mv 2022-09
dc.type.none.fl_str_mv info:eu-repo/semantics/article
info:eu-repo/semantics/publishedVersion
http://purl.org/coar/resource_type/c_6501
info:ar-repo/semantics/articulo
format article
status_str publishedVersion
dc.identifier.none.fl_str_mv http://hdl.handle.net/11336/211604
Albani, Clara Maria; Borgo, Jimena; Fabbri, Julia; Pensel, Patricia Eugenia; Fasciani, L.; et al.; Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s; Oxford University Press; Evidence-Based Complementary and Alternative Medicine; 2022; 9-2022; 1-10
1741-427X
1741-4288
CONICET Digital
CONICET
url http://hdl.handle.net/11336/211604
identifier_str_mv Albani, Clara Maria; Borgo, Jimena; Fabbri, Julia; Pensel, Patricia Eugenia; Fasciani, L.; et al.; Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.s; Oxford University Press; Evidence-Based Complementary and Alternative Medicine; 2022; 9-2022; 1-10
1741-427X
1741-4288
CONICET Digital
CONICET
dc.language.none.fl_str_mv eng
language eng
dc.relation.none.fl_str_mv info:eu-repo/semantics/altIdentifier/url/https://www.hindawi.com/journals/ecam/2022/6371849/
info:eu-repo/semantics/altIdentifier/doi/10.1155/2022/6371849
dc.rights.none.fl_str_mv info:eu-repo/semantics/openAccess
https://creativecommons.org/licenses/by-nc-sa/2.5/ar/
eu_rights_str_mv openAccess
rights_invalid_str_mv https://creativecommons.org/licenses/by-nc-sa/2.5/ar/
dc.format.none.fl_str_mv application/pdf
application/pdf
application/pdf
application/pdf
application/pdf
dc.publisher.none.fl_str_mv Oxford University Press
publisher.none.fl_str_mv Oxford University Press
dc.source.none.fl_str_mv reponame:CONICET Digital (CONICET)
instname:Consejo Nacional de Investigaciones Científicas y Técnicas
instname_str Consejo Nacional de Investigaciones Científicas y Técnicas
reponame_str CONICET Digital (CONICET)
collection CONICET Digital (CONICET)
repository.name.fl_str_mv CONICET Digital (CONICET) - Consejo Nacional de Investigaciones Científicas y Técnicas
repository.mail.fl_str_mv dasensio@conicet.gov.ar; lcarlino@conicet.gov.ar
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spelling Antiparasitic Effects of Asteraceae Species Extracts on Echinococcus granulosus s.sAlbani, Clara MariaBorgo, JimenaFabbri, JuliaPensel, Patricia EugeniaFasciani, L.Elso, Orlando GermanPapademetrio, Daniela LauraGrasso, Daniel HectorPaladini, A.Beer, Maria FlorenciaFarias, Nahuel EmilianoElissondo, N.Gambino, G.Zoppi, J.Sülsen, Valeria PatriciaElissondo, María CelinaAsteraceaeEchinococcus granulosusCystic echinococcosishttps://purl.org/becyt/ford/3.3https://purl.org/becyt/ford/3Cystic echinococcosis is a zoonotic disease caused by the parasite Echinococcus granulosus sensu lato (s.l.), which is worldwide distributed and causes long-lasting infections in animals and humans. The existing treatment is limited to the use of benzimidazoles, mainly albendazole (ABZ). However, it has unwanted side effects and its efficacy is about 50%. The Asteraceae family includes plants that have therapeutic applications (medicinal species) and has an important role in new drug development. The species belonging to a different genus of this family show a wide range of anti-inflammatory, antimicrobial, antioxidant, hepatoprotective, and antiparasitic activities, among others. The aim of the present study was to evaluate the in vitro efficacy of extracts of four Asteraceae species against protoscoleces of E. granulosus sensu stricto (s.s.). On the other hand, the Stevia aristata extract was assessed on the murine cyst of E. granulosus (s.s.) and the efficacy of S. aristata extract was investigated in a murine model of CE. Stevia satureiifolia, S. aristata, Grindelia pulchella, and G. chiloensis extracts at 100 μg/mL caused a decrease in protoscoleces viability; however, S. aristata extract produced the greatest in vitro protoscolicidal effect. After 20 days of treatment with the highest concentration (100 μg/mL) of S. aristata extract, protoscoleces viability decreased to 0%. The tegumental changes observed by scanning electron microscopy were consistent with the reduction in vitality. The collapse of the germinal layer was registered in 60 ± 5.8% and 83.3 ± 12.0% of cysts treated during 4 days with 50 and 100 μg/ml, respectively. The half maximal effective concentration (EC50) value of the S. aristata extract against E. granulosus (s.s.) cysts was 47.86 μg/mL (96 h). The dosage of infected animals with the 50 mg kg-1 dose of S. aristata extract resulted in a significant reduction in cyst weight in comparison with the control group. In conclusion, S. aristata extract was demonstrated to exert a marked effect, both in vitro and in the murine model.Fil: Albani, Clara Maria. Universidad Nacional de Mar del Plata. Instituto de Investigaciones En Produccion, Sanidad y Ambiente. - Consejo Nacional de Investigaciones Cientificas y Tecnicas. Centro Cientifico Tecnologico Conicet - Mar del Plata. Instituto de Investigaciones En Produccion, Sanidad y Ambiente.; Argentina. Universidad Nacional de Mar del Plata. Facultad de Ciencias Exactas y Naturales. Departamento de Biología. Laboratorio de Zoonosis Parasitarias; ArgentinaFil: Borgo, Jimena. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Departamento de Farmacología. Cátedra de Farmacognosia; Argentina. Consejo Nacional de Investigaciones Científicas y Técnicas. Oficina de Coordinación Administrativa Houssay. Instituto de Química y Metabolismo del Fármaco. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Instituto de Química y Metabolismo del Fármaco; ArgentinaFil: Fabbri, Julia. Universidad Nacional de Mar del Plata. Facultad de Ciencias Exactas y Naturales. Departamento de Biología. Laboratorio de Zoonosis Parasitarias; Argentina. Universidad Nacional de Mar del Plata. Facultad de Cs.exactas y Naturales. Instituto de Investigaciones En Sanidad Produccion y Ambiente. - Comision de Investigaciones Cientificas de la Provincia de Buenos Aires. Instituto de Investigaciones En Sanidad Produccion y Ambiente.; ArgentinaFil: Pensel, Patricia Eugenia. Universidad Nacional de Mar del Plata. Facultad de Cs.exactas y Naturales. Instituto de Investigaciones En Sanidad Produccion y Ambiente. - Comision de Investigaciones Cientificas de la Provincia de Buenos Aires. Instituto de Investigaciones En Sanidad Produccion y Ambiente.; ArgentinaFil: Fasciani, L.. Universidad Nacional de Mar del Plata. Facultad de Ciencias Exactas y Naturales. Departamento de Biología. Laboratorio de Zoonosis Parasitarias; ArgentinaFil: Elso, Orlando German. Consejo Nacional de Investigaciones Científicas y Técnicas. Oficina de Coordinación Administrativa Houssay. Instituto de Química y Metabolismo del Fármaco. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Instituto de Química y Metabolismo del Fármaco; Argentina. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Departamento de Farmacología. Cátedra de Farmacognosia; ArgentinaFil: Papademetrio, Daniela Laura. Consejo Nacional de Investigaciones Científicas y Técnicas. Oficina de Coordinación Administrativa Houssay. Instituto de Estudios de la Inmunidad Humoral Prof. Ricardo A. Margni. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Instituto de Estudios de la Inmunidad Humoral Prof. Ricardo A. Margni; ArgentinaFil: Grasso, Daniel Hector. Consejo Nacional de Investigaciones Científicas y Técnicas. Oficina de Coordinación Administrativa Houssay. Instituto de Estudios de la Inmunidad Humoral Prof. Ricardo A. Margni. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Instituto de Estudios de la Inmunidad Humoral Prof. Ricardo A. Margni; ArgentinaFil: Paladini, A.. Universidad Nacional de La Plata. Facultad de Ciencias Veterinarias. Cátedra de Parasitología y Enfermedades Parasitarias; ArgentinaFil: Beer, Maria Florencia. Consejo Nacional de Investigaciones Científicas y Técnicas. Oficina de Coordinación Administrativa Houssay. Instituto de Química y Metabolismo del Fármaco. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Instituto de Química y Metabolismo del Fármaco; ArgentinaFil: Farias, Nahuel Emiliano. Consejo Nacional de Investigaciones Científicas y Técnicas. Centro Científico Tecnológico Conicet - Mar del Plata. Instituto de Investigaciones Marinas y Costeras. Universidad Nacional de Mar del Plata. Facultad de Ciencias Exactas y Naturales. Instituto de Investigaciones Marinas y Costeras; ArgentinaFil: Elissondo, N.. No especifíca;Fil: Gambino, G.. No especifíca;Fil: Zoppi, J.. No especifíca;Fil: Sülsen, Valeria Patricia. Consejo Nacional de Investigaciones Científicas y Técnicas. Oficina de Coordinación Administrativa Houssay. Instituto de Química y Metabolismo del Fármaco. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Instituto de Química y Metabolismo del Fármaco; Argentina. Universidad de Buenos Aires. Facultad de Farmacia y Bioquímica. Departamento de Farmacología. Cátedra de Farmacognosia; ArgentinaFil: Elissondo, María Celina. Universidad Nacional de Mar del Plata. Facultad de Cs.exactas y Naturales. Instituto de Investigaciones En Sanidad Produccion y Ambiente. - Comision de Investigaciones Cientificas de la Provincia de Buenos Aires. 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