Bioinspired Functional Catechol Derivatives through Simple Thiol Conjugate Addition

The combination of the surface-adhesive properties of catechol rings and functional moieties conveying specific properties is very appealing to materials chemistry, but the preparation of catechol derivatives often requires elaborate synthetic routes to circumvent the intrinsic reactivity of the cat...

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Detalles Bibliográficos
Autores: Mancebo Aracil, Juan, Casagualda, Carolina, Moreno Villaecija, Miguel Angel, Nador, Fabiana Gabriela, García Pardo, Javier, Franconetti García, Antonio, Busqué, Félix, Alibés, Ramón, Esplandiu, María José, Ruiz Molina, Daniel, Sedó Vegara, Josep
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2019
País:Argentina
Institución:Consejo Nacional de Investigaciones Científicas y Técnicas
Repositorio:CONICET Digital (CONICET)
Idioma:inglés
OAI Identifier:oai:ri.conicet.gov.ar:11336/120483
Acceso en línea:http://hdl.handle.net/11336/120483
Access Level:acceso abierto
Palabra clave:BIOINSPIRED MATERIALS
CATECHOLS
FUNCTIONAL COATINGS
SULFUR
SURFACES AND INTERFACES
THERANOSTICS
THIOL CONJUGATE ADDITION
https://purl.org/becyt/ford/1.4
https://purl.org/becyt/ford/1
Descripción
Sumario:The combination of the surface-adhesive properties of catechol rings and functional moieties conveying specific properties is very appealing to materials chemistry, but the preparation of catechol derivatives often requires elaborate synthetic routes to circumvent the intrinsic reactivity of the catechol ring. In this work, functional catechols are synthesized straightforwardly by using the bioinspired reaction of several functional thiols with o-benzoquinone. With one exception, the conjugated addition of the thiol takes place regioselectively at the 3-position of the quinone, and is rationalized by DFT calculations. Overall, this synthetic methodology provides a general and straightforward access to functional and chain-extended catechol derivatives, which are later tested with regard to their hydro-/oleophobicity, colloidal stability, fluorescence, and metal-coordinating capabilities in proof-of-concept applications.