Synthesis of D-homo analogs of neurosteroids

17(13→18)-Abeo and D-homo analogs of the natural neurosteroid 3α-hydroxy-5αH-pregnan-20-one were prepared by anionic or radical (mercury (II) hydride mediated) rearrangements of steroidal cyclopropylketones respectively.

Detalles Bibliográficos
Autores: Di Chenna, P., Ghini, A.A., Burton, G.
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2000
País:Argentina
Institución:Universidad Nacional de Buenos Aires. Facultad de Ciencias Exactas y Naturales
Repositorio:Biblioteca Digital (UBA-FCEN)
Idioma:inglés
OAI Identifier:paperaa:paper_14203049_v5_n3_p447_DiChenna
Acceso en línea:http://hdl.handle.net/20.500.12110/paper_14203049_v5_n3_p447_DiChenna
Access Level:acceso abierto
Palabra clave:11alpha hydroxyprogesterone
3alpha hydroxy 5alpha pregnan 20 one derivative
cyclopropylketone derivative
dehydropregnenolone acetate
ketone derivative
mercury derivative
neurosteroid derivative
pregnenolone derivative
steroid
unclassified drug
conference paper
drug structure
drug synthesis
reaction analysis
Descripción
Sumario:17(13→18)-Abeo and D-homo analogs of the natural neurosteroid 3α-hydroxy-5αH-pregnan-20-one were prepared by anionic or radical (mercury (II) hydride mediated) rearrangements of steroidal cyclopropylketones respectively.