Extracellular signal-regulated kinase phosphorylates tumor necrosis factor alpha-converting enzyme at threonine 735: a potential role in regulated shedding.

[EN]The ectodomain of certain transmembrane proteins can be released by the action of cell surface proteases, termed secretases. Here we have investigated how mitogen-activated protein kinases (MAPKs) control the shedding of membrane proteins. We show that extracellular signal-regulated kinase (Erk)...

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Detalles Bibliográficos
Autores: Díaz Rodríguez, María Elena, Montero González, Juan Carlos, Esparís Ogando, Azucena, Yuste, Laura, Pandiella Alonso, Atanasio
Tipo de recurso: artículo
Estado:Versión publicada
Fecha de publicación:2002
País:España
Institución:Universidad de Salamanca (USAL)
Repositorio:GREDOS. Repositorio Institucional de la Universidad de Salamanca
OAI Identifier:oai:gredos.usal.es:10366/167830
Acceso en línea:http://hdl.handle.net/10366/167830
Access Level:acceso abierto
Palabra clave:TACE, Cleavage, MAPKs
Retroviridae
Binding Sites
Transfection
Restriction Mapping
Humans
HeLa Cells
Metalloendopeptidases
Amino Acid Sequence
Carrier Proteins
Membrane Proteins
Mitogen-Activated Protein Kinases
Tetradecanoylphorbol Acetate
Phosphorylation
Threonine
Protein Kinase C
ADAM Proteins
2302 Biochemistry
proteína cinasa C
mapeo por restricción
humanos
treonina
proteínas transportadoras
células HeLa
proteína cinasas activadas por mitógenos
acetato de tetradecanoilforbol
sitios de unión
transfección
metaloendopeptidasas
proteínas ADAM
secuencia de aminoácidos
proteínas de membranas
fosforilación
Descripción
Sumario:[EN]The ectodomain of certain transmembrane proteins can be released by the action of cell surface proteases, termed secretases. Here we have investigated how mitogen-activated protein kinases (MAPKs) control the shedding of membrane proteins. We show that extracellular signal-regulated kinase (Erk) acts as an intermediate in protein kinase C-regulated TrkA cleavage. We report that the cytosolic tail of the tumor necrosis factor alpha-converting enzyme (TACE) is phosphorylated by Erk at threonine 735. In addition, we show that Erk and TACE associate. This association is favored by Erk activation and by the presence of threonine 735. In contrast to the Erk route, the p38 MAPK was able to stimulate TrkA cleavage in cells devoid of TACE activity, indicating that other proteases are also involved in TrkA shedding. These results demonstrate that secretases are able to discriminate between the different stimuli that trigger membrane protein ectodomain cleavage and indicate that phosphorylation by MAPKs may regulate the proteolytic function of membrane secretases.