Dehydrogenative [2 + 2 + 2] Cycloaddition of Cyano-yne-allene Substrates: Convenient Access to 2,6-Naphthyridine Scaffolds

A rhodium-catalyzed [2 + 2 + 2] cycloaddition of cyano-yne-allene scaffolds followed by a dehydrogenative process enabling the direct synthesis of unsaturated pyridine-containing compounds that can be conveniently converted to 2,6-naphthyridine derivatives is reported

Detalhes bibliográficos
Autores: Haraburda, Ewelina, Lledó Ponsati, Agustí, Roglans i Ribas, Anna, Pla i Quintana, Anna
Formato: artículo
Estado:Versión aceptada para publicación
Fecha de publicación:2015
País:España
Recursos:Varias* (Consorci de Biblioteques Universitáries de Catalunya, Centre de Serveis Científics i Acadèmics de Catalunya)
Repositorio:Recercat. Dipósit de la Recerca de Catalunya
OAI Identifier:oai:recercat.cat:10256/10958
Acesso em linha:http://hdl.handle.net/10256/10958
Access Level:acceso abierto
Palavra-chave:Reaccions d'addició
Addition reactions
Catàlisi
Catalysis
Catalitzadors de rodi
Rhodium catalyst
Rodi
Rhodium
Ciclització (Química)
Ring formation (Chemistry)
Descrição
Resumo:A rhodium-catalyzed [2 + 2 + 2] cycloaddition of cyano-yne-allene scaffolds followed by a dehydrogenative process enabling the direct synthesis of unsaturated pyridine-containing compounds that can be conveniently converted to 2,6-naphthyridine derivatives is reported